彭俊梅｜南华大学｜学者主页

2025

关于8种含氮杂环光催化合成的研究进展（英文）

刘艺琦，陈文婕，赵泽艳，王苏棋，唐圣松，何卫民，彭俊梅

《有机化学》

2024

High affinity and low PARP-trapping benzimidazole derivatives as a potential warhead for PARP1 degraders.

Xiaoyu Peng, Yang Li, Junfeng Qu, Lizhi Jiang, Kaiyue Wu, Dan Liu, Yuping Chen, Junmei Peng, Yu Guo, Xuan Cao

European journal of medicinal chemistry

DOI

2023

基于OBE教学理念的药物化学教学改革探索

杨泽华，谢志忠，唐国涛，彭俊梅，杨晓燕，伍造端

《广州化工》

2023

The Progress of Small Molecule Targeting BCR-ABL in the Treatment of Chronic Myeloid Leukemia.

Yuan Zhang, Xin Wu, Xueyan Sun, Jun Yang, Chang Liu, Guo-Tao Tang, Xiao-Yong Lei, Honglin Huang, Junmei Peng

Mini-Reviews in Medical Chemistry

DOI

2023

Design, synthesis, and evaluation of 1H‐benzo[d]imidazole‐4‐carboxamide PARP‐1 inhibitors using different saturated nitrogen‐contained heterocycle as linker group

Kai-Yue Wu, Xiaoyu Peng, Yang Li, Miao Chen, Yun-feng Liu, Liu Dan, Lizhi Jiang, He Yan, Junmei Peng, Xuan Cao

Chemical Biology and Drug Design

DOI

2022

探索药学专业课程思政深化“三全育人”

贺冬秀，喻翠云，雷小勇，彭俊梅，刘阳，王卫国

《卫生职业教育》

2022

电化学促进的五元芳香杂环与硫氰酸铵氧化交叉脱氢偶联反应（英文）

李红霞，陈棚，伍智林，陆雨函，彭俊梅，陈锦杨，何卫民

《有机化学》

2022

新时代药学专业学位研究生导师队伍建设探索

贺冬秀，喻翠云，彭俊梅，雷小勇，李兰芳，刘阳

《创新创业理论研究与实践》

2022

电催化肼、丙二酮和2-溴丙二酸二乙酯三组分合成4-溴吡唑

穆思宇，李红霞，伍智林，彭俊梅，陈锦杨，何卫民

《有机化学》

2022

染料木素锌、铜金属配合物的制备及抗癌活性研究

王有娣，彭俊梅，刘铭美，徐娟娟

《大豆科学》

2022

Recent Progress of the research on the benzimidazole PARP-1 inhibitors.

Kai-Yue Wu, Miao Chen, Xiaoyu Peng, Yang Li, Guo-Tao Tang, Junmei Peng, Xuan Cao

Mini-Reviews in Medical Chemistry

DOI

2022

Applications of "linkers" in fragment-based drug design.

Xin Wu, Yuan Zhang, Songbin Liu, Chang Liu, Guo-Tao Tang, Xuan Cao, Xiao-Yong Lei, Junmei Peng

Bioorganic chemistry (Print)

DOI

2022

Recent progress of research on anti‐tumor agents using benzimidazole as the structure unit

Kai-Yue Wu, Xiaoyu Peng, Miao Chen, Yang Li, Guo-Tao Tang, Junmei Peng, Yuan-Yuan Peng, Xuan Cao

Chemical Biology and Drug Design

DOI

2022

Advances in Development of Drugs for Chronic Myelogenous Leukemia.

Yuan Zhang, Xin Wu, Xueyan Sun, Jun Yang, Chang Liu, Guo-Tao Tang, Xiao-Yong Lei, Honglin Huang, Junmei Peng

Mini-Reviews in Medical Chemistry

DOI

2021

以白藜芦醇为结构单元的丹酚酸A类似物的合成及其体外抗氧化作用测定

陈妙佳，马思明，李洋，贺芬，彭俊梅，唐国涛，曹轩

《中南医学科学杂志》

DOI

2021

Design, synthesis, and biological evaluation of 3′,4′,5′‐trimethoxy evodiamine derivatives as potential antitumor agents

Yijiao Peng, Runde Xiong, Zhen Li, Junmei Peng, Zhi-Zhong Xie, Xiao-Yong Lei, D. He, Guo-Tao Tang

Drug development research (Print)

DOI

2021

Discovery of a Potential Multi-Target Anti-Tumor Agent via Structural Modification on Flavonoid

Xiang-Ping Deng, Yang-Yang Zou, Renbo Liu, Yijiao Peng, Chenglin Ouyang, Junmei Peng, Xiao-Yong Lei, Zhi-Zhong Xie, Chong Li, Guo-Tao Tang

Polycyclic aromatic compounds (Print)

DOI

2021

Anti-chronic myeloid leukemia activity and quantitative structure-activity relationship of novel thiazole aminobenzamide derivatives.

Yuan Zhang, Juan Liu, Xin Wu, Suming Yang, Yao-Wang Li, Songbin Liu, Saifei Zhu, Xuan Cao, Zhi-Zhong Xie, Xiao-Yong Lei, Honglin Huang, Junmei Peng

Bioorganic & Medicinal Chemistry Letters

DOI

2021

Synthesis and evaluation of 2‐(4‐[4‐acetylpiperazine‐1‐carbonyl] phenyl)‐1H‐benzo[d]imidazole‐4‐carboxamide derivatives as potential PARP‐1 inhibitors and preliminary study on structure‐activity relationship

Miao Chen, Honglin Huang, Kaiyue Wu, Yun-feng Liu, Lizhi Jiang, Yang Li, Guo-Tao Tang, Junmei Peng, Xuan Cao

Drug development research (Print)

DOI

2020

基于“雨课堂”的“药物化学实验”课程教学模式改革实践

刘映，李帑洛，郭玉，彭俊梅，贺冬秀

《教育教学论坛》

2020

仪器分析在线教学实践与思考

刘阳，刘运美，曾要富，彭俊梅，郭玉

《广州化工》

2020

Recent advances in Bcr‐Abl tyrosine kinase inhibitors for overriding T315I mutation

Juan Liu, Yuan Zhang, Honglin Huang, Xiao-Yong Lei, Guo-Tao Tang, Xuan Cao, Junmei Peng

Chemical Biology and Drug Design

DOI

2019

基于Topomer CoMFA法的类黄酮类化合物乙酰胆碱酯酶抑制剂的三维定量构效关系研究

李曼玉，杨梅芳，刘美香，姚旭，彭俊梅，刘映

《化学世界》

DOI

2019

Design, synthesis and broad-spectrum Bcr-Abl inhibitory activity of novel thiazolamide–benzamide derivatives

Juan Liu, Honglin Huang, Xiang-Ping Deng, Runde Xiong, Xuan Cao, Guo-Tao Tang, Xin Wu, Shi-juan Xu, Junmei Peng

RSC Advances

DOI

2019

Design, synthesis and biological evaluation of tryptamine salicylic acid derivatives as potential antitumor agents.

Runde Xiong, D. He, Xiang-Ping Deng, Juan Liu, Xiao-Yong Lei, Zhi-Zhong Xie, Xuan Cao, Yanming Chen, Junmei Peng, Guo-Tao Tang

MedChemComm

DOI

2019

Anti-proliferative activity and structure-activity relationship of honokiol derivatives.

Ding-Yan Lin, Zhong-Zhong Yan, Ai-Yu Chen, Jiao Ye, Ai-Xi Hu, Juan Liu, Junmei Peng, Xiao-Yun Wu

Bioorganic & Medicinal Chemistry

DOI

2019

FS-7 inhibits MGC-803 cells growth in vitro and in vivo via down-regulating glycolysis.

Xiang-Ping Deng, Zhong-Li Li, Runde Xiong, Juan Liu, Renbo Liu, Junmei Peng, Yanming Chen, Xiao-Yong Lei, Xuan Cao, Xing Zheng, Zhi-Zhong Xie, Guo-Tao Tang

Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie

DOI

2018

阿魏酸酰胺类乙酰胆碱酯酶抑制剂的三维定量构效关系研究

刘映，谢秀珍，李曼玉，杨梅芳，刘美香，周珂，彭俊梅，姚旭

《广州化工》

2018

碱性条件下合成3-羧基苯基硫脲的初步探讨

张鑫鑫，刘娟，刘映，罗景顺，陈垚，李澳，彭俊梅

《广东化工》

2018

依托协同创新平台加强构建研究型药学实验课程体系

刘映，彭俊梅，姚旭，丁岚，李帑洛，唐国涛，贺冬秀，涂剑

《广州化工》

2018

有机药物波谱解析教学改革探讨

刘阳，杨寒幸，刘运美，彭俊梅，贺冬秀

《药学教育》

2018

Semi-synthesis, structural modification and biological evaluation of 5-arylbenzofuran neolignans

Ding-Yan Lin, Long Wang, Zhong-Zhong Yan, Jiao Ye, Ai-Xi Hu, Hong-Dong Liao, Juan Liu, Junmei Peng

RSC Advances

DOI

2017

正交实验法优化碧螺春茶叶中总黄酮提取工艺

刘映，王敏，谢秀珍，彭俊梅，唐国涛

《应用化工》

2017

药物化学互动式网络教学改革探索

贺冬秀，喻翠云，李兰芳，彭俊梅，唐国涛，陈洪飞

《教育教学论坛》

2017

药学专业《仪器分析》课程教学改革探索

刘阳，贺艳，刘运美，彭俊梅，郭玉

《广州化工》

2017

Synthesis and antitumor activity of novel N-(5-benzyl-4-(tert-butyl)thiazol-2-yl)-2-(piperazin-1-yl)acetamides

Zhi-Lin Wu, Na Ding, Yu-Ting Tang, Jiao Ye, Junmei Peng, Ai-Xi Hu

Research on chemical intermediates (Print)

DOI

2016

药学专业《分析化学》课程的信息化教学改革初探

刘阳，刘运美，彭俊梅，郭玉

《医学教育研究与实践》

2016

浅谈如何提高药学专业学生学习有机药物波谱解析的兴趣

彭俊梅，刘映，刘运美，刘阳，唐国涛

《广东化工》

2015

《药事管理学》课程的信息化教学改革探索

贺冬秀，喻翠云，唐国涛，彭俊梅，刘映，谢志忠

《教育教学论坛》

2015

基于上转换纳米材料的pH传感器研究

刘映，胡益辉，彭俊梅

《科技资讯》

2015

Design, synthesis and neuraminidase inhibitory activity of N-(5-benzyl-4-(tert-butyl)thiazol-2-yl)benzamides

Zhi-Lin Wu, Junmei Peng, Ai-Xi Hu, Jiao Ye, Guo-Xi Li

Medicinal Chemistry Research

DOI

2014

Synthesis,Crystal Structure and Antitumor Activity of N-(4-tert-butyl-5-(4-chlorobenzyl)thiazol-2-yl)-2,6-difluorobenzamide

申坤，彭俊梅，李婉，颜晓维，胡艾希

Chinese Journal of Structural Chemistry

2014

Synthesis and antitumor activity of 4-tert-butyl-5-benzyl-2-benzyliminothiazoles

Jiao Ye, Shen-Yi Qiu, Ai-Xi Hu, Junmei Peng, Zhi-Hui Qin

Chemical Research in Chinese Universities

DOI

2013

4-烷基-6-芳基-1,3-噻嗪的合成与生物活性

Wan-Shui Li, Ai-Xi Hu, Ailin Liu, Junmei Peng, Lin Xia, Wei-Qing Tan

DOI

2013

基于4,4-二甲基-1-芳基-1-戊烯-3-酮的噻唑及嘧啶衍生物的合成与生物活性

彭俊梅

《湖南大学》

2013

5-苄基-4-叔丁基-2-芳氨基噻唑氢溴酸盐的合成、表征及抗肿瘤活性

彭俊梅，李婉，申坤，霍素芳，叶姣，胡艾希

《高等学校化学学报》

2013

4-(7-Methoxy-2,2-dimethyl-2,3-dihydrobenzo-furan-5-yl)-N-(pyridin-2-yl)thiazol-2-amine: Chiral Crystal from Achiral Molecule

彭俊梅，曹高，罗先福，胡艾希，叶姣，欧晓明

Chinese Journal of Structural Chemistry

2013

Design and Synthesis of 4‐Alkyl‐2‐amino(acetamino)‐6‐aryl‐1,3‐thiazine Derivatives as Influenza Neuraminidase Inhibitors

Wan Li, Lin Xia, Ai-Xi Hu, Ai-Lin Liu, Junmei Peng, Wei-Qing Tan

Archiv der Pharmazie

DOI

2012

Synthesis, Crystal Structure and Antitumor Activity of 4-tert-Butyl-N-(2-fluorophenyl)-5- (1H-1,2,4-triazol-1-yl)-thiazol-2-amine

李婉，叶姣，沈芳，彭俊梅，胡艾希

Chinese Journal of Structural Chemistry

2011

鱼藤酮肟羧酸酯的合成和生物活性

叶姣，彭俊梅，胡艾希，王超，邹孟，欧晓明

《有机化学》

2010

4-(N-乙酰氨基)-3-(4-芳基噻唑-2-氨基)苯甲酸乙酯的合成与生物活性

夏林，胡艾希，彭俊梅

《有机化学》

2007

Ethyl 2‐methyl‐1‐(4‐phenylthiazol‐2‐yl)‐1H‐benzimidazole‐6‐carboxylate

Li-Min He, Ai-Xi Hu, Gao Cao, Junmei Peng

DOI

精选作品

期刊论文

关于8种含氮杂环光催化合成的研究进展（英文）

High affinity and low PARP-trapping benzimidazole derivatives as a potential warhead for PARP1 degraders.

基于OBE教学理念的药物化学教学改革探索

The Progress of Small Molecule Targeting BCR-ABL in the Treatment of Chronic Myeloid Leukemia.

Design, synthesis, and evaluation of 1H‐benzo[d]imidazole‐4‐carboxamide PARP‐1 inhibitors using different saturated nitrogen‐contained heterocycle as linker group

探索药学专业课程思政 深化“三全育人”

电化学促进的五元芳香杂环与硫氰酸铵氧化交叉脱氢偶联反应（英文）

新时代药学专业学位研究生导师队伍建设探索

电催化肼、丙二酮和2-溴丙二酸二乙酯三组分合成4-溴吡唑

染料木素锌、铜金属配合物的制备及抗癌活性研究

Recent Progress of the research on the benzimidazole PARP-1 inhibitors.

Applications of "linkers" in fragment-based drug design.

Recent progress of research on anti‐tumor agents using benzimidazole as the structure unit

Advances in Development of Drugs for Chronic Myelogenous Leukemia.

以白藜芦醇为结构单元的丹酚酸A类似物的合成及其体外抗氧化作用测定

Design, synthesis, and biological evaluation of 3′,4′,5′‐trimethoxy evodiamine derivatives as potential antitumor agents

Discovery of a Potential Multi-Target Anti-Tumor Agent via Structural Modification on Flavonoid

Anti-chronic myeloid leukemia activity and quantitative structure-activity relationship of novel thiazole aminobenzamide derivatives.

Synthesis and evaluation of 2‐(4‐[4‐acetylpiperazine‐1‐carbonyl] phenyl)‐1H‐benzo[d]imidazole‐4‐carboxamide derivatives as potential PARP‐1 inhibitors and preliminary study on structure‐activity relationship

基于“雨课堂”的“药物化学实验”课程教学模式改革实践

仪器分析在线教学实践与思考

Recent advances in Bcr‐Abl tyrosine kinase inhibitors for overriding T315I mutation

基于Topomer CoMFA法的类黄酮类化合物乙酰胆碱酯酶抑制剂的三维定量构效关系研究

Design, synthesis and broad-spectrum Bcr-Abl inhibitory activity of novel thiazolamide–benzamide derivatives

Design, synthesis and biological evaluation of tryptamine salicylic acid derivatives as potential antitumor agents.

Anti-proliferative activity and structure-activity relationship of honokiol derivatives.

FS-7 inhibits MGC-803 cells growth in vitro and in vivo via down-regulating glycolysis.

阿魏酸酰胺类乙酰胆碱酯酶抑制剂的三维定量构效关系研究

碱性条件下合成3-羧基苯基硫脲的初步探讨

依托协同创新平台加强构建研究型药学实验课程体系

有机药物波谱解析教学改革探讨

Semi-synthesis, structural modification and biological evaluation of 5-arylbenzofuran neolignans

正交实验法优化碧螺春茶叶中总黄酮提取工艺

药物化学互动式网络教学改革探索

药学专业《仪器分析》课程教学改革探索

Synthesis and antitumor activity of novel N-(5-benzyl-4-(tert-butyl)thiazol-2-yl)-2-(piperazin-1-yl)acetamides

药学专业《分析化学》课程的信息化教学改革初探

浅谈如何提高药学专业学生学习有机药物波谱解析的兴趣

《药事管理学》课程的信息化教学改革探索

基于上转换纳米材料的pH传感器研究

Design, synthesis and neuraminidase inhibitory activity of N-(5-benzyl-4-(tert-butyl)thiazol-2-yl)benzamides

Synthesis,Crystal Structure and Antitumor Activity of N-(4-tert-butyl-5-(4-chlorobenzyl)thiazol-2-yl)-2,6-difluorobenzamide

Synthesis and antitumor activity of 4-tert-butyl-5-benzyl-2-benzyliminothiazoles

4-烷基-6-芳基-1,3-噻嗪的合成与生物活性

基于4,4-二甲基-1-芳基-1-戊烯-3-酮的噻唑及嘧啶衍生物的合成与生物活性

5-苄基-4-叔丁基-2-芳氨基噻唑氢溴酸盐的合成、表征及抗肿瘤活性

4-(7-Methoxy-2,2-dimethyl-2,3-dihydrobenzo-furan-5-yl)-N-(pyridin-2-yl)thiazol-2-amine: Chiral Crystal from Achiral Molecule

Design and Synthesis of 4‐Alkyl‐2‐amino(acetamino)‐6‐aryl‐1,3‐thiazine Derivatives as Influenza Neuraminidase Inhibitors

Synthesis, Crystal Structure and Antitumor Activity of 4-tert-Butyl-N-(2-fluorophenyl)-5- (1H-1,2,4-triazol-1-yl)-thiazol-2-amine

鱼藤酮肟羧酸酯的合成和生物活性

4-(N-乙酰氨基)-3-(4-芳基噻唑-2-氨基)苯甲酸乙酯的合成与生物活性

Ethyl 2‐methyl‐1‐(4‐phenylthiazol‐2‐yl)‐1H‐benzimidazole‐6‐carboxylate

会议论文

5-苄基-4-叔丁基-2-芳氨基噻唑的合成及其抑制人癌细胞增殖作用

1,3-噻嗪类流感病毒NAIs的设计、合成及其生物活性研究

1,3-噻嗪类化合物的合成及其应用

探索药学专业课程思政深化“三全育人”