Kecheng Yang, Wentao Yang, Longwei Guo, Xin-Yu Wang, Hongmin Liu, Xiao-Quan Feng, Yuefeng Bi, Xiao-Le Chen, Xu Gao (2026). Co-Folding-Driven Structural Mapping of Reversible LSD1 Inhibitors Reveals Unexplored Chemical Space and Binding Diversity. Journal of Chemical Information and Modeling.DOI
Yalnaz Naseem, Jianshu Dong, Kecheng Yang, Cong Han, Xinli Ma, Jian Li, Syed Azeem, Hongmin Liu (2026). Structure-Guided Discovery of Isoindolinone–Triazolopyrimidine Hybrids as Potential Skp1–Skp2 Inhibitors: Integrated Docking, Molecular Dynamics, and Machine learning modelling. In Silico Research in Biomedicine.DOI
Shuo Yuan, Yi-Ru Bai, Ruifang Li, Jian Song, Tingting Liu, Sai‐Yang Zhang, Hong‐Min Liu, Ying Xu (2026). Silver-Catalyzed Cascade Reactions for the Synthesis of Indopyran Pseudo-Natural Products as Potent Anti-tumor Agents. Organic Letters.DOI
Kaizhao Hu, Kun Zhang, Rui-Hao Chui, Wenhui Qiu, Pei-Pei Miao, Linlin Zhang, Meng Ding, Qingjin Zhang, Bing Zhao, Xiao-Jing Shi, Hongmin Liu (2025). Molecular hybridization strategy - discovery of 2,3-diarylpyrazine derivatives as potent Skp2 inhibitors with improved anti-tumor activity and enhanced cisplatin sensitivity. European journal of medicinal chemistry.DOI
Xin-Hui Zhang, Huiqin Kang, Bing-Qian Li, Yuhan Xiong, Shuxian Zheng, Di Zhang, Yuan-Fan Liu, Shi-Yu Li, Ying Liu, Hongmin Liu, Ya Gao, Li-Ying Ma (2025). Structural Optimization of 1,3-Diaryl-1,2,4-triazole-Capped Histone Deacetylase 6 Inhibitors to Obtain Novel Antiesophageal Cancer Candidates. Journal of Medicinal Chemistry.DOI
H. M. Akram, Yu-Lin Liu, Jianshu Dong, Xue-Ke Zhao, Li-Dong Wang, Wen Zhao, Hongmin Liu, LiYing Ma, Cong Han (2025). Discovery of W478, a novel SHMT2 inhibitor for the treatment of esophageal carcinoma. Bioorganic chemistry (Print).DOI
Shuqi Lou, Yingying Huang, Xiaohui Wang, Ying-Mei Li, Feifan Li, Leyi Ma, Yu Zhou, Hongmin Liu, Ling Fu, Yuefeng Bi (2025). Hepatoprotective effects of the active extracts from Chrysanthemi Indici Flos via regulating epigenetic networks. Fitoterapia.DOI
Mengzhen Li, Woonghee Kim, Han Jin, Hong Yang, Xiang-Tai Kong, Xi-Ya Song, Hasan Turkez, Yuefeng Bi, Chengxue Pan, Ling Fu, Hongmin Liu, M. Uhlén, Cheng Zhang, Adil Mardinoğlu (2025). Anticancer effects and mechanisms of Pulsatilla chinensis, Bupleurum chinense and Polyporus umbellatus on human lung carcinoma and hepatoma cells. Computational and Structural Biotechnology Journal.DOI
Nigatu Tadesse, Manni He, Juan Li, Hong‐Min Liu (2025). Challenges of folate species analysis in food and biological matrices by liquid chromatography-tandem mass spectrometery. Bioanalysis.DOI
Ya Gao, Haiqian Nie, Hong‐Min Liu, Xinhui Zhang, Liying Ma (2025). Rational Design, Synthesis, and Biological Assessment of Potential Indole‐Capped HDAC6 Inhibitors for Gastric Cancer Suppression. MedComm.DOI
yanzhi wang, Shanshan Sun, Mengqian Liu, Sai Zhang, Jiaxin Zheng, Hong‐Min Liu (2025). Glycyrrhetinic Acid-Biguanide Conjugate-Based Nanoparticles as a Multi-Functional Drug Delivery System: Paclitaxel Encapsulation and Targeted Therapy. Molecular Pharmaceutics.DOI
Xing‐Jie Dai, Leipeng Xue, Ying Liu, Shuwu Wang, Ying Li, Jiayi Yin, Hao-Zhe Long, Huimin Liu, Ning Wang, Guo‐Liang Lu, Yan Li, Hong‐Min Liu, Bo Wang, Yi‐Chao Zheng (2025). Identification of Novel Phenoxazine-Derived LSD1 Inhibitors Suppressing Gastric Cancer Stemness by β-Catenin Transcriptional Regulation. Journal of Medicinal Chemistry.DOI
Han Jiahui, Wang Shihao, Hongjing Chen, Gu Dongling, Zichen Yang, Hao Wang, Fuqiang Yu, Lingling Chi, Yu Ke, Hong‐Min Liu, Zhang Qiurong (2025). Design, Synthesis, and Antitumor Activity Evaluation of Novel 2,4,7-Trisubstituted Quinazoline Derivatives Containing an Aminomethyl Piperidine Moiety. Russian Journal of Bioorganic Chemistry.DOI
Xin Yang, Xiang Li, Yuelin Zhang, Shengnan Zhang, Miao Zhang, Chong Sun, Li Yang, Hong‐Min Liu, Shuo Yuan (2024). Targeting undruggable protein KRAS for cancer therapy: novel opportunities and challenges. Future Medicinal Chemistry.DOI
Xueming Li, Fenglian Zhang, Yu Ke, Hong‐Min Liu, Zhenbo Hu, Zhenbo Hu, Liuya Wei (2024). Differentiation of Acute Leukemia Cells Including Cells with MLL-AF4 Rearrangements Induced by Jiyuan Oridonin A. Recent Patents on Anti-Cancer Drug Discovery.DOI
Shihao Wang, Zichen Yang, Dongling Gu, Jiahui Han, Hongjing Chen, Hao Wang, Jiaxin Zheng, Hong‐Min Liu, Yu Ke, Qiurong Zhang (2024). Design, synthesis, and evaluation of antitumor activity of quinazoline derivatives containing different terminal segments of basic amine groups. Medicinal Chemistry Research.DOI
Dandan Shen, Yuelin Zhang, Xiang Li, Yi‐Ru Bai, Jun‐Feng Xiong, Dong‐Jie Seng, Yao‐Dong Zhang, Hong‐Min Liu, Shuo Yuan, Li Yang (2024). The mechanism of action and chemical synthesis of FDA newly approved drug molecules. Drug Development Research.DOI
Yi‐Ru Bai, Wei‐Guang Yang, Rui Jia, Ju‐Shan Sun, Dandan Shen, Hong‐Min Liu, Shuo Yuan (2024). The recent advance and prospect of poly(ADP‐ribose) polymerase inhibitors for the treatment of cancer. Medicinal Research Reviews.DOI
Yi‐Ru Bai, Dong‐Jie Seng, Ying Cao Xu, Yaodong Zhang, Wenjuan Zhou, Yang-Yang Jia, Jian Zheng Song, Zhangxu He, Hong‐Min Liu, Shuo Yuan (2024). A comprehensive review of small molecule drugs approved by the FDA in 2023: Advances and prospects. European Journal of Medicinal Chemistry.DOI
Moges Dessale Asmamaw, Ang He, Lirong Zhang, Hong‐Min Liu, Ya Gao (2024). Histone deacetylase complexes: Structure, regulation and function. Biochimica et Biophysica Acta (BBA) - Reviews on Cancer.DOI
Juan Li, Wenchao Hu, Mengxue Liu, Yingqi Tian, Manni He, Hong‐Min Liu (2024). Simultaneous determination of folic acid photolysis products and oxidized guanine derivatives in plasma by liquid chromatography‐tandem mass spectrometry. Journal of Separation Science.DOI
Yajie Liu, Yajie Liu, Pengxing He, Xubin Ma, Ying-qi Tian, Yu Zhang, Yang Wang, Yingjie Jia, Hong‐Min Liu, Ying Liu, Ying Liu, Yichao Xu (2024). The combination of SLC7A11 inhibitor and oridonin synergistically inhibits cervical cancer cell growth by decreasing the NADPH/NADP+ ratio. Genes & Diseases.DOI
Ning-Jie Guo, Bo Wang, Yu Zhang, Huiqin Kang, Haiqian Nie, Meng-Kai Feng, Xi-Ya Zhang, Lijuan Zhao, Ning Wang, Hong‐Min Liu, Yi‐Chao Zheng, Wen J. Li, Ya Gao (2024). USP7 as an emerging therapeutic target: A key regulator of protein homeostasis. International Journal of Biological Macromolecules.DOI
Liang Shen, Bo Wang, Shaopeng Wang, Shi‐Kun Ji, Meng‐Jie Fu, Shuwu Wang, Wenqing Hou, Xing‐Jie Dai, Hong‐Min Liu (2024). Combination Therapy and Dual-Target Inhibitors Based on LSD1: New Emerging Tools in Cancer Therapy. Journal of Medicinal Chemistry.DOI
Hang Xie, Jian-Jia Liang, Yalei Wang, Tianxing Hu, Jinyi Wang, Ruihua Yang, Jun-Ke Yan, Qiurong Zhang, Xia Xu, Hong‐Min Liu, Yu Ke (2020). The design, synthesis and anti-tumor mechanism study of new androgen receptor degrader. European Journal of Medicinal Chemistry.DOI
Yang Zhang, Luye Zhang, Limin Liu, Tao Wang, Yaqi Meng, Na Li, Erdong Li, Zhengjie Wang, Xiujuan Liu, Jiaxin Zheng, Lihong Shan, Hong‐Min Liu, Qiurong Zhang (2020). Synthesis and Antitumor Activity Evaluation of Novel Hydrazone-Substituted Pyrimidine Derivatives. Chinese Journal of Organic Chemistry.DOI
Zhiru Wang, Wen-Ting Kang, Yinghua You, Jing‐Ru Pang, Hongmei Ren, Zhenhe Suo, Hong‐Min Liu, Yi‐Chao Zheng (2019). USP7: Novel Drug Target in Cancer Therapy. Frontiers in Pharmacology.DOI
Juan Li, Qingli Wang, Yi‐Chao Zheng, Piao Zhou, Xia Xu, Xueqi Liu, Longfei Zhao, Hong‐Min Liu (2019). Development of a mass spectrometry-based pseudotargeted metabolomics strategy to analyze hormone-stimulated gastric cancer cells. Journal of Pharmaceutical and Biomedical Analysis.DOI
Jianwei Zhao, Zeng-Hui Wu, Jia–Wen Guo, Ming-Jie Huang, Ya-Zhen You, Hong‐Min Liu, Li‐Hua Huang (2019). Synthesis and anti-gastric cancer activity evaluation of novel triazole nucleobase analogues containing steroidal/coumarin/quinoline moieties. European Journal of Medicinal Chemistry.DOI
Jianwei Zhao, Jia–Wen Guo, Ming-Jie Huang, Ya-Zhen You, Zeng-Hui Wu, Hong‐Min Liu, Li‐Hua Huang (2019). Design, synthesis and biological evaluation of new steroidal β-triazoly enones as potent antiproliferative agents. Steroids.DOI
Er-dong Li, Lin Qiao, Yaqi Meng, Lu-ye Zhang, Panpan Song, Na Li, Jingchao Xin, Peng Yang, Chongnan Bao, Dan-qing Zhang, Yang Zhang, Ji-kuan Wang, Qiurong Zhang, Hong‐Min Liu (2019). 2,4-Disubstituted quinazolines targeting breast cancer cells via EGFR-PI3K. European Journal of Medicinal Chemistry.DOI
Juan Li, Qingli Wang, Piao Zhou, Qiqi Fan, Tianze Cao, Yatong Li, Mengxuan Li, Zhang Yue, Mengfei Bian, Hongmin Liu (2018). Development of LC-MS-based pseudotargeted metabolomics method and its application in hormone-stimulated MGC803 Cells. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Yunkai Shi, Wenjuan Zhou, Yu Liu, Jingjing Song, Yanyan Que, Wen Zhao, Bin Yu, Hongmin Liu (2018). Discovery of a potent inhibitor of DCN1-UBC12 interaction. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Piao Zhou, Qiqi Fan, Juan Li, Mengchen An, Hongmin Liu (2018). Establishment and application of 23 kinds of nucleosides and modified nucleosides in cell samples. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Na Li, Jingchao Xin, Yaqi Meng, Erdong Li, Chongnan Bao, Peng Yang, Jiaxin Zheng, Qiurong Zhang, Hongmin Liu (2018). Design and synthesis of novel 2,4,6-substituted pyrimidine derivatives as potential antitumor agents. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Zhangxu He, Chen Liu, Yi Ying Wang, Liying Ma, Hongmin Liu (2018). Design,synthesis,and structure-activity relationship of novel pan HDAC inhibitors based on indole. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Jingchao Xin, Na Li, Erdong Li, Yaqi,Meng, Jiaxin,Zheng, Qiurong Zhang, Hongmin Liu (2018). The design,synthesis and antitumor activity of novel tetrazolo[5,1-a]phthalazine derivatives. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Qianqian Liang, Hao Zhang, Liyan Zhou, Bing Zhao, Hongmin Liu (2018). Design synthesis and bioactivity evaluation of quinoline KDM5B inhibitors. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Qisheng Ma, Yinghua You, Xingyu Ma, Qian li, Tongtong Li, Zhiyang Ruan, Zhiling Chen, Yichao Zheng, Bin Yu, Hongmin Liu (2018). Design,synthesis and biological evaluation of indolines as potent lysine specific demethylase 1(LSD1/KDM1A) inhibitors. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Yaqi Meng, Erdong Li, Na Li, Jingchao Xin, Chongnan Bao, Peng Yang, Jiaxin Zheng, Qiurong Zhang, Hongmin Liu (2018). USP7:a promising target for cancer therapy. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Feifei Yang, Liying Ma, Hongmin Liu (2018). Design,synthesis and biological evaluation of novel indole-based hybrids. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Shuai Wang, Lijie Zhao, Kai Tang, Xiaojing Shi, Lina Ding, Yichao Zheng, Bin Yu, Hongmin Liu (2018). The development of small molecules targeting DCN1-UBC12 protein-protein interactions. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Li Zhu, Xue An, Peipei Gao, Lihong Shan, Hongmin Liu (2018). Design and synthesis of 15β,16β-methylene steroid-2-benzylidene-4,6-diene-3,17-dione derivatives. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Maksim Semenov, Yuan Shuo, Lingyu Li, Bin Yu, Hongmin Liu, Wen Zhao (2018). Structure-based discovery and optimization of new potent and selective BET inhibitors for potential treatment of heart failure. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Yanan Li, YuANDi Zhao, Peng Yang, Linlin Lou, Yiying Wang, Chen Liu, Qingyuan Wei, Hongmin Liu (2018). Design and synthesis of novel 6-chloro-purine-based derivatives as potential selective anti-lung cancer agents. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Jianjia Liang, Hang Xie, Ruihua Yang, Longfei Zhao, Ying Liu, Yu Ke, Hongmin Liu (2018). A "Click Chemistry Platform" for the rapid synthesis of small-molecule-mediated degradation of the androgen receptor. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Yuandi Zhao, Bo Wang, Yanan Li, Liying Ma, Hongmin Liu (2018). Design,synthesis of novel 1,2,3-triazoles and derivatives as potential IDO1 inhibitors. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Yandan Ren, Mengying Zhang, Yang Wang, Tianli Fan, Qi Zhao, Yu Zhao, Hongmin Liu, Guiqin Hou, Zhaoming Lu (2018). FLI-06 suppresses proliferation,induces apoptosis and cell cycle arrest by targeting LSD1 and Notch pathway in esophageal squamous cell carcinoma cells. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Xiaojing Shi, Xiaojing Li, Yi Huang, Jun Dong, Hongmin Liu (2018). Characterize the expression of Skp2 in gastric carcinoma:promotion of tumorigenesis. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Ying Liu, Longfei Zhao, Jianjia Liang, Zhusong Cao, Xiaojing Li, Le Yang, Bo Wang, Fengzhi Suo, Jinyi Wang, Ruihua Yang, Yu Ke, Liying Ma, Hongmin Liu (2018). Design,synthesis and in vitro activity of novel triazine-based LSD1 inhibitors. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Zhongrui Li, Fengzhi Suo, DANDan Shen, Shuo Yuan, Bin Yu, Yichao Zheng, Hongmin Liu (2018). Identification of natural protoberberine alkaloids as potent,selective,and cellular active LSD1/KDM1A inhibitors for AML treatment. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Dandan Shen, Shuai Wang, Qimeng Song, Yichao Zheng, Hongmin Liu (2018). Establishment of screening platform for small molecular inhibitors of BRD4 and screening and activity evaluation of inhibitors. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Yichao Zheng, Hongmin Liu (2018). Interruption of a paracrine amplification loop between LSD1 and TGF β1 by LSD1 inhibitor. 《第11届世界华人药物化学研讨会(ISCMC 2018)》.
Ting Ma, Wenjun Peng, Lisha Zhao, Ruyue Wang, Qian Wang, Yanqin Tu, Hongmin Liu (2018). Polyphyllin G induced apoptosis and protective autophagy by targeting MAPK pathway in colorectal carcinoma cells. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Tiantian Qin, Dongxiao Yang, Xueyan Zhang, Leilei Li, Weihua Liu, Junfeng Huo, Xiaoli Shi, Cong Wang, Hongmin Liu (2018). ASC26,a Selective ABCB1 inhibitor reverses ABCB1-mediated drug resistance in cancer cells. 《第11届世界华人药物化学研讨会(ISCMC 2018)》.
Zhenya Wang, Xiaoning Hu, Xiaodong Mou, Congcong Wang, Yuanyuan Li, Xinli Chen, Yayun Tan, Chunli Wu, Hongmin Liu, Haiwei Xu (2018). Design,synthesis and anti-virus activity of a novel butenolide as inhibitors of neuraminidase from influenza A virus H1N1 in vitro and in Vivo. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Yaquan Cao, Bing Zhao, Lingling Ren, Qinyan Shi, Yunan Su, Hongmin Liu (2018). Histone demethylase KDM5B. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Shuo Yuan, Si-Xi Wang, Tongtong Li, Jie Zhang, Qiangyan Zhang, Wen Zhao, Bin Yu, Hongmin Liu (2018). Design and synthesis of potent and selective BRD4 inhibitors. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Shuo Yuan, Dandan Shen, Jinjie Chen, Zixin Qiu, Yonggang Liu, Yichao Zheng, Bin Yu, Hongmin Liu (2018). Brφnsted acid-catalyzed direct C(sp2)-H activation enabling the discovery of biaryl compounds as novel BRD4 inhibitors. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Kai Tang, Bin Yu, Hongmin Liu (2018). Discovery of new tetrahydroisoquinoline-based LSD1/KDM1A inhibitors from natural product Higenamine. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Peng Yang, Yanan Li, Yuanzi Zhao, Qiurong Zhang, Linlin Lou, Qingyuan Wei, Chen Liu, Yiying Wang, Hongmin Liu (2018). Design,synthesis and biological evaluation of imidazo[4,5-c]pyridine derivatives as potential antitumor agents. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Qiuhua Zhang, Bin Yu, Hongmin Liu (2018). Structure-based design of KDM5A/B protein degraders. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Erdong Li, Yaqi Meng, Jingchao Xin, Na Li, Chongnan Bao, Peng Yang, Peirong Zhao, Qiurong Zhang, Hongmin Liu (2018). Design and synthesis of novel 2,4,5-trisubstituted quinazoline derivatives. 《第11届世界华人药物化学研讨会(ISCMC 2018)论文摘要集》.
Qisheng Ma, Yongfang Yao, Yi‐Chao Zheng, Siqi Feng, Junbiao Chang, Bin Yu, Hong‐Min Liu (2018). Ligand-based design, synthesis and biological evaluation of xanthine derivatives as LSD1/KDM1A inhibitors. European Journal of Medicinal Chemistry.DOI
Yu Ke, Jian-Jia Liang, Rui-Juan Hou, Mingming Li, Longfei Zhao, Wancong Wang, Ying Liu, Hang Xie, Ruihua Yang, Tianxing Hu, Jinyi Wang, Hong‐Min Liu (2018). Synthesis and biological evaluation of novel Jiyuan Oridonin A-1,2,3-triazole-azole derivatives as antiproliferative agents. European Journal of Medicinal Chemistry.DOI
Yong‐Gang Hua, Qian‐Qian Yang, Yi Yang, Mei‐Jing Wang, Wen-Chao Chu, Peng-Yan Bai, De-Yun Cui, En Zhang, Hong‐Min Liu (2018). Metal-free synthesis of 1,2-amino alcohols by one-pot olefin aziridination and acid ring-opening. Tetrahedron Letters.DOI
Yong‐Gang Hua, Lan‐Ping Han, Qian‐Qian Yang, Mei‐Jing Wang, En Zhang, Hong‐Min Liu (2018). A Practical and Efficient Stereoselective Synthesis of (S)‐Rivastigmine and (R)‐Rivastigmine. ChemistrySelect.DOI
Yunkai Shi, Bo Wang, Xiaoli Shi, Yuandi Zhao, Bin Yu, Hong‐Min Liu (2018). Synthesis and biological evaluation of new steroidal pyridines as potential anti-prostate cancer agents. European Journal of Medicinal Chemistry.DOI
Wen Li, Lina Ding, Hong‐Min Liu, Qidong You (2017). Synthesis, biological evaluation, and molecular docking of ropivacaine analogs as local anesthetic agents. Medicinal Chemistry Research.DOI
Peng-Fei Geng, Congcong Wang, Zhonghua Li, Xiaoning Hu, Taoqian Zhao, Dong‐Jun Fu, Bing Qiang Zhao, Bin Yu, Hong‐Min Liu (2017). Design, synthesis and preliminary biological evaluation of 5,8-dihydropteridine-6,7-diones that induce apoptosis and suppress cell migration. European Journal of Medicinal Chemistry.DOI
Zhonghua Li, Taoqian Zhao, Xue‐qi Liu, Bing Qiang Zhao, Chao Wang, Peng Geng, Yaquan Cao, Dong‐Jun Fu, Liping Jiang, Bin Yu, Hong‐Min Liu (2017). Synthesis and preliminary antiproliferative activity of new pteridin-7(8H)-one derivatives. European Journal of Medicinal Chemistry.DOI
Zhonghua Li, Xue‐Qi Liu, Taoqian Zhao, Peng Geng, Wen-Ge Guo, Bin Yu, Hong‐Min Liu (2017). Design, synthesis and preliminary biological evaluation of new [1,2,3]triazolo[4,5- d ]pyrimidine/thiourea hybrids as antiproliferative agents. European Journal of Medicinal Chemistry.DOI
Zhonghua Li, Xue‐Qi Liu, Taoqian Zhao, Peng-Fei Geng, Ying Liu, Bing Qiang Zhao, Wen-Ge Guo, Bin Yu, Hong‐Min Liu (2017). Design, synthesis and preliminary antiproliferative activity studies of new diheteroaryl thioether derivatives. Bioorganic & Medicinal Chemistry Letters.DOI
Dong‐Jun Fu, Ruo-Han Zhao, Jiahuan Li, Jiajia Yang, Ruo-Wang Mao, Bowen Wu, Ping Li, Xiaolin Zi, Qingqing Zhang, Huijie Cai, Sai‐Yang Zhang, Yanbing Zhang, Hong‐Min Liu (2017). Molecular diversity of phenothiazines: design and synthesis of phenothiazine–dithiocarbamate hybrids as potential cell cycle blockers. Molecular Diversity.DOI
Zhong-Hua Li, Xue‐Qi Liu, Peng Geng, Ji Zhang, Jinlian Ma, Bo Wang, Taoqian Zhao, Bing Qiang Zhao, Xinhui Zhang, Bin Yu, Hong‐Min Liu (2017). Design, synthesis and antiproliferative activity of thiazolo[5,4-d]pyrimidine derivatives through the atom replacement strategy. European Journal of Medicinal Chemistry.DOI
Dong‐Jun Fu, Jian Song, Yuhui Hou, Ruo-Han Zhao, Jiahuan Li, Ruo-Wang Mao, Jiajia Yang, Ping Li, Xiaolin Zi, Zhonghua Li, Qingqing Zhang, Feiyan Wang, Sai‐Yang Zhang, Yanbing Zhang, Hong‐Min Liu (2017). Discovery of 5,6-diaryl-1,2,4-triazines hybrids as potential apoptosis inducers. European Journal of Medicinal Chemistry.DOI
Panpan Song, Fei Cui, Na Li, Jingchao Xin, Qisheng Ma, Xiangchuan Meng, Chaojie Wang, Qinpo Cao, Yifei Gu, Yu Ke, Qiurong Zhang, Hong‐Min Liu (2017). Synthesis, Cytotoxic Activity Evaluation of Novel 1,2,3‐Triazole Linked Quinazoline Derivatives. Chinese Journal of Chemistry.DOI
Feng‐Wu Liu, Wenke Xu, Hui Yang, Yingju Liu, Yingchun Hua, Bin He, Xin Ning, Zhiyan Qin, Hong‐Min Liu (2017). Facile Approaches to 2-Deoxy-d-glucose and 2-Deoxy-α-d-glucopyranonucleosides from d-Glucal. Synthesis.DOI
Kezheng Peng, Yu Ke, Qi Zhao, Fei Tian, Hong‐Min Liu, Guiqin Hou, Zhaoming Lu (2017). OP16, a novel ent-kaurene diterpenoid, potentiates the antitumor effect of rapamycin by inhibiting rapamycin-induced feedback activation of Akt signaling in esophageal squamous cell carcinoma. Biochemical Pharmacology.DOI
Cong Wang, Liubin Guo, Saiqi Wang, Junwei Wang, Yongmei Li, Yinhui Dou, Ran Wang, Hongge Shi, Yu Ke, Hong‐Min Liu (2017). Anti-proliferative effect of Jesridonin on paclitaxel-resistant EC109 human esophageal carcinoma cells. International Journal of Molecular Medicine.DOI
Biao Hu, Bo Wang, Bing Qiang Zhao, Qian Guo, Zhonghua Li, Xinhui Zhang, Guang-Yao Liu, Ying Liu, Ying Chun Tang, Fan Luo, Ya Nan Du, Yaxin Chen, Liying Ma, Hong‐Min Liu (2017). Thiosemicarbazone-based selective proliferation inactivators inhibit gastric cancer cell growth, invasion, and migration. MedChemComm.DOI
Zhonghua Li, Xue‐Qi Liu, Peng Geng, Jinlian Ma, Taoqian Zhao, Hao-Ming Wei, Bin Yu, Hong‐Min Liu (2017). Design, synthesis, and biological evaluation of new thiazolo[5,4-d]pyrimidine derivatives as potent antiproliferative agents. MedChemComm.DOI
Yong-Cheng Ma, Yu Ke, X. Zi, Fei Zhao, Lin Yuan, Ying-Ming Zhu, Xia-Xia Fan, N. Zhao, Qiao-Yan Li, Yu-Hua Qin, Hongmin Liu (2016). Induction of the mitochondria-mediated apoptosis in human esophageal cancer cells by DS2, a newly synthetic diterpenoid analog, is regulated by Bax and caused by generation of reactive oxygen species. OncoTarget.DOI
Fu‐Qiang Wang, Hui Yang, Bin He, Yong‐Kang Jia, Shi‐Yao Meng, Chao Zhang, Hong‐Min Liu, Feng‐Wu Liu (2016). ChemInform Abstract: A Novel Domino Approach for Synthesis of Indolyl Tetrahydropyrano[4,3‐c]pyrazole Derivatives as Anticancer Agents. ChemInform.DOI
Xiaojing Shi, Lina Ding, Wenjuan Zhou, Yage Ji, Junwei Wang, Huimin Wang, Yong‐Cheng Ma, Guozhong Jiang, Kai Tang, Yu Ke, Wen Zhao, Hong‐Min Liu (2016). Pro-Apoptotic Effects of JDA-202, a Novel Natural Diterpenoid, on Esophageal Cancer Through Targeting Peroxiredoxin I. Antioxidants and Redox Signaling.DOI
En Zhang, Wei-Wei Jiao, Shang Wang, Jinmei Xu, Xiaojing Shi, Yanchao Wang, Yana Wang, Hong‐Min Liu (2016). Design, synthesis, and preliminary evaluation of the biological activity of dithiocarbamate-3-epi-jaspine B hybrids. Medicinal Chemistry Research.DOI
Fu-Qiang Wang, Hui Yang, Bin He, Yong‐Kang Jia, Shi‐Yao Meng, Chao Zhang, Hong‐Min Liu, Feng‐Wu Liu (2016). A novel domino approach for synthesis of indolyl tetrahydropyrano[4,3-c]pyrazole derivatives as anticancer agents. Tetrahedron.DOI
Wenjuan Zhou, Liying Ma, Biao Hu, Lingyu Li, Bo Wang, Hong‐Min Liu, Wen He Zhao (2016). Abstract 3813: Potent compounds targeting the human MutT homolog 1 (hMTH1) activity and their cytotoxicity evaluation. Cancer Research.DOI
Lihong Shan, Yang Li, Yanjie Chen, Minghui Yin, Jiajia Huang, Zhenzhong Zhang, Xiufang Shi, Hong‐Min Liu (2016). Microbial hydroxylation of 17β-estradiol by Penicillium brevicompactum. Biocatalysis and Biotransformation.DOI
Lihong Shan, Kai Jiao, Minghui Yin, Jiajia Huang, Yanjie Chen, Shangshang Qin, Hong‐Min Liu (2016). Biotransformation of 5-en-3β-ol steroids byMucor circinelloides lusitanicus. Biocatalysis and Biotransformation.DOI
Yanling Zhang, Yafei Li, Junwei Wang, Bin Yu, Yunkai Shi, Hong‐Min Liu (2016). Multicomponent assembly of novel antiproliferative steroidal dihydropyridinyl spirooxindoles. Steroids.DOI
Juan Li, Yu Chen, Yanyan Diao, Yingqian Su, Qingli Wang, Zhicun Yao, Tianxiang Yi, Wenting Jin, Dan Yang Zhao, Caihong Wang, Mengru Liu, Hong‐Min Liu (2016). Identification of metabolites of the novel anti‐tumor drug candidate MDH‐7 in rat urine by liquid chromatography coupled with triple quadrupole linear ion trap mass spectrometry. Rapid Communications in Mass Spectrometry.DOI
En Zhang, Hong‐Min Liu, Shang Wang, Jie Gao, Xiaojing Shi, Mingming Wang, Shuai-Min Xu (2016). Synthesis and Evaluation of the Antitumor Activities of Two Series of Jaspine B Analogues Bearing 2-Alkyloxymethyl Group. Heterocycles.DOI
Bin Yu, De‐Quan Yu, Hong‐Min Liu (2015). ChemInform Abstract: Spirooxindoles: Promising Scaffolds for Anticancer Agents. ChemInform.DOI
Yanling Zhang, Yafei Li, Yunkai Shi, Bin Yu, Guochen Zhang, Ping‐Ping Qi, Dong‐Jun Fu, Lihong Shan, Hong‐Min Liu (2015). Efficient three-component one-pot synthesis of steroidal polysubstituted anilines. Steroids.DOI
Bin Yu, Zhiqiang Yu, Ping‐Ping Qi, De‐Quan Yu, Hong‐Min Liu (2015). ChemInform Abstract: Discovery of Orally Active Anticancer Candidate CFI‐400945 Derived from Biologically Promising Spirooxindoles: Success and Challenges. ChemInform.DOI
Bei-Xi Jia, Qian-Qian Huangfu, Feng‐Xiao Ren, Lu Jia, Yanbing Zhang, Hong‐Min Liu, Jie Yang, Wang Qiang (2014). Identification and quantification of flavonoids and chromes inBaeckea frutescensby using HPLC coupled with diode-array detection and quadruple time-of-flight mass spectrometry. Natural Product Research.DOI
Qiu‐Rong Zhang, Deng‐Qi Xue, Peng He, Kun‐Peng Shao, Peng‐Ju Chen, Yifei Gu, Jingli Ren, Lihong Shan, Hong‐Min Liu (2014). ChemInform Abstract: Synthesis and Antimicrobial Activities of Novel 1,2,4‐Triazolo[3,4‐a]phthalazine Derivatives. ChemInform.DOI
Xu Henan, Lan Zhang, Hong‐Min Liu, Sijie Liu, Huangquan Lin, Yan Wang, David Chi‐Cheong Wan, Chun Hu (2013). Synthesis, characterization and biological activity of 3-aryl-6-(4-fluorobenzyl)-7H-thiazolo[3,2-b]-1,2,4-triazin-7-one derivatives as novel acetylcholinesterase inhibitors. Rare & Special e-Zone (The Hong Kong University of Science and Technology).
Qiurong Zhang, Peng He, Guangqiang Zhou, Kang Yu, Hong‐Min Liu (2013). 4-Cyclopropyl-1-(6′-deoxy-1′,2′-O-isopropylidene-α- D -glucofuranosyl)-1H-1,2,3-triazole. Acta Crystallographica Section E Structure Reports Online.DOI
Bin Yu, En Zhang, Yuan Fang, Xiaonan Sun, Jingli Ren, De‐Quan Yu, Hong‐Min Liu (2013). ChemInform Abstract: The New Convenient Synthesis of Novel γ‐Alkylidenebutenolides from 6‐Aminopenicillanic Acid. ChemInform.DOI
Haiwei Xu, Pingjuan Jiang, Weiyi Li, Junfeng Wang, Hong‐Min Liu (2011). Synthesis and Bioactivities of Andrographolide Derivatives: New (−)‐Limonidilactone Analogues. Chinese Journal of Chemistry.DOI
Xiaojuan Wang, Haiwei Xu, Linlin Guo, En Zhang, Guang‐Wei Chen, Xiao Ping Guo, Hong‐Min Liu (2011). ChemInform Abstract: Synthesis of Various Substituted Spiro‐ and Bicyclethiazolidine‐2‐thiones by a Multicomponent Reaction and Biological Evaluation in vitro. ChemInform.DOI
Jingyu Zhang, Xuehui Hou, Hong‐Min Liu (2011). Synthesis, Crystal Structure and Hydrolysis of a Novel Anhydrogalactosucrose: 2′‐Methoxyl‐O‐1′,4′:3′,6′‐dianhydro‐β‐D‐fructofuranosyl 3,6‐anhydro‐4‐chloro‐4‐deoxy‐α‐D‐galactopyranoside. Chinese Journal of Chemistry.DOI
Li‐Hua Huang, Yanguang Wang, Gong Xu, Xiang-Hua Zhang, Yong‐Fei Zheng, Hui-Li He, Wenzheng Fu, Hong‐Min Liu (2011). Novel 4-azasteroidal N-glycoside analogues bearing sugar-like D ring: Synthesis and anticancer activities. Bioorganic & Medicinal Chemistry Letters.DOI
Qiurong Zhang, Xuebin Chen, Nan Zhu, Tengfei Jiang, Hong‐Min Liu (2011). 3,5-Di-O-benzoyl-1,2-O-isopropylidene-α- D -ribo-hexos-3-ulo-1,4:3,6-difuranose. Acta Crystallographica Section E Structure Reports Online.DOI
Qiurong Zhang, Pan Li, Xuebin Chen, Xiandong Wang, Hong‐Min Liu (2011). 3,6-Didehydro-5-hydroxy-1,2-O-isopropylidene-5-C-nitromethyl-α- D -glucofuranose. Acta Crystallographica Section E Structure Reports Online.DOI
Qiurong Zhang, Chunli Wu, Pengyun Li, Weiyan Cheng, Hong‐Min Liu (2011). N-Benzyl-6-deoxy-3,6-iminomethylene-1,2,3,5-O-tetraacetyl-α- D -1(S)-epiallofuranose. Acta Crystallographica Section E Structure Reports Online.DOI
Hong Shu Liu, Fuyi Zhang, Jinpeng Li, Xuebin Yan, Hong‐Min Liu, Yufen Zhao (2011). Novel Methyl 4,6-O-benzylidene-3-ketoglucopyranosid-fused γ-lactam: Synthesis and Crystal Structure. Journal of Chemical Crystallography.DOI
Hai-Yan Zhang, Tian-Zeng Zhao, Yue Zhou Wei, Hong‐Min Liu (2011). Two new sesquiterpene polyol esters from the root barks ofCelastrus angulatus. Journal of Asian Natural Products Research.DOI
Heping Li, Yu Peng, Hongjie Zhang, Hong‐Min Liu (2008). ChemInform Abstract: Synthesis of 5‐Androstene‐3β,7α,17β‐triol and 5‐Androstene‐3β,7β,17β‐triol. ChemInform.DOI
Yanbing Zhang, Piyong Zhang, Gui‐Fu Dai, Hong‐Min Liu (2008). ChemInform Abstract: Study on the Synthesis and Bioactivity of Novel Mahkoside A Derivatives. ChemInform.DOI
Hong‐Min Liu (2008). Synthesis of 7α-OH-Dehydroepiandrosterone and Evaluation of Its Bioactivity. Zhōnghuá yàoxué zázhì.
Haiwei Xu, Jianye Zhang, Hong‐Min Liu, Jun‐Feng Wang (2006). Synthesis of Andrographolide Cyclophosphate Derivatives and Their Antitumor Activities. ChemInform.DOI
Gui‐Fu Dai, Haiwei Xu, Junfeng Wang, Feng‐Wu Liu, Hong‐Min Liu (2006). Studies on the Novel α‐Glucosidase Inhibitory Activity and Structure—Activity Relationships for Andrographolide Analogues. ChemInform.DOI
Hong‐Min Liu, Feng‐Wu Liu, Dapeng Zou, Gui‐Fu Dai (2005). Asymmetric Synthesis of Novel Tetrahydroquinoline Derivatives with a Sugar Building Block and Their Bioactivities. ChemInform.DOI
WU Chun-li, Qiurong Zhang, Shan Li-hong, Yankai Liu, Hong‐Min Liu (2005). Improved synthesis of danofloxacin. Zhongguo yaowu huaxue zazhi.
Hong‐Min Liu, Fuyi Zhang, Dapeng Zou (2003). Stereoselective Synthesis of 2,2‐Bis(C‐Branched‐Chain)glucopyranosid‐3‐ulose via an Autoxidation—Michael Addition Reaction. ChemInform.DOI
李雯,刘宏民(2002). 对位取代苯酚氧甙类化合物的相转移催化合成与结构表征. 《有机化学》.
Fuyi Zhang, Chenxia Du, Hong‐Min Liu, Yu Zhu (2002). ChemInform Abstract: A Novel Glycoside Lactone Derivative with a 2‐C‐Unsaturated Diester Substituent. ChemInform.DOI
预印本
Yi‐Chao Zheng, Jingru Pang, Yu Zhang, Hao Zhu, Dandan Shen, Bo Wang, Yan Li, Guo‐Liang Lu, Ning Wang, Zheng-Hong Yang, Xin Dai, Hong‐Min Liu (2026). Targeting LSD1 inhibits gastric cancer by reprogramming macrophages and restoring T-cell response. Research Square.DOI
Liying Ma, Xinhui Zhang, Haiqian Nie, Junru Zhao, Mengkai Feng, Xiaoqian Yu, Yulin Liu, Huiqin Kang, Yuanfan Liu, Shiyu Li, Hong‐Min Liu, Ya Gao (2025). Design, Synthesis and Biological Evaluation of Novel Indole-Capped Histone Deacetylase 6 Inhibitors as Anti-Gastric Cancer Agents. SSRN Electronic Journal.DOI
Liying Ma, Xinhui Zhang, Haiqian Nie, Junru Zhao, Mengkai Feng, Yulin Liu, Huiqin Kang, Yuanfan Liu, Shiyu Li, Hong‐Min Liu, Ya Gao (2025). Design, Synthesis and Biological Evaluation of Novel Histone Deacetylase 6 Inhibitors Containing Indole-Based Cap Groups. SSRN Electronic Journal.DOI
Linyue Bai, Liang Shen, Qianqian Zhang, Zhuang Hu, Yanjun Tang, Mengjie Fu, Hong‐Min Liu, Xing‐Jie Dai, Siqi Feng (2024). Accelerating Small Molecule Ferroptosis Regulator Development with Advances in Biological Functions.DOI
yanzhi wang, Linchao Wang, H.M. Chang, qing shen, sai zhang, Shanshan Sun, Ying Liu, Jiaxin Zheng, Hong‐Min Liu (2023). Enhancing anti-tumor therapy with agmatine-cholesterol conjugate liposomes: in vitro and in vivo evidence. Research Square.DOI
Xiaojie Si, Fuqiang Yu, Hao Wang, Lingling Chi, Honglin Dai, Chao Gao, Yingnan Zhu, Hong‐Min Liu, Qiurong Zhang (2023). Design, synthesis and antitumor activity evaluation in vitro of 4,6,7-trisubstituted quinazoline derivatives containing acrylamide moiety. Research Square.DOI