2026
Discovery of Novel HPK1 Inhibitors via Chemistry-Based Direct-to-Bioassay Screening and SAR Optimization
Yiping Duan, Chen He, Zhichao Guo, Kai Sun, Tiandong Zheng, Yang Lu, Baixue Zhang, Wenyi Zhong, Yansong Ren, Jie Liu, Shengtao Xu, Jinyi Xu
Journal of Medicinal Chemistry