刘祈星｜三峡大学｜学者主页

2026

基于CVL-231的环丁胺类M4正向变构调节剂的设计、合成与活性

李馥莼，李文歆，何姝芳，陈毅昆，周皓，周海峰，刘祈星，田峦鸢

《高等学校化学学报》

2026

新型N-2,3-二氟苯基环丁胺类M4 AChR正向变构调节剂的设计、合成与活性

刘敏，陈毅昆，田峦鸢，周海峰，周皓，刘祈星

《有机化学》

2026

新型噻唑烷酮三氟乙基亚砜类化合物的设计、合成及杀螨活性

张世稳，蔡胜梅，陈锦彪，刘祈星，周海峰

《农药学学报》

DOI

2026

Mechanochemical NH 4 Cl-mediated hydrogen-bonding network reconstruction of HFIP: enabling yne-allylic substitutions

Qianzhi Yang, Xuguang Kong, Xin Liu, Qixing Liu, Linhong Zuo, Haifeng Zhou

Chemical Communications

DOI

2026

Nickel-Catalyzed Asymmetric Hydrogenation of All-Carbon Tetrasubstituted Alkenes Enabled by van der Waals Interactions.

Cong-Cong Yin, Zichang Wang, Yuli Liang, Jia-Mu Deng, Yunxin Zheng, Qixing Liu, Jie Zeng, Xu-Meng Zhang, Hai-Feng Zhou

Angewandte Chemie

DOI

2025

盐酸曲美他嗪的合成工艺改进

陈敏，陈多鹏，刘祈星，刘义稳，周海峰

《中国医药工业杂志》

2025

含螺噻唑烷酮的三氟乙基硫醚类化合物的合成与杀螨活性

熊文敏，陈锦彪，包如胜，林健，田平义，刘祈星，周海峰

《农药学学报》

2025

利格列汀原料药有关物质的合成

丑瑞龙，章华，游珊，刘祈星，周海峰

《中国药学杂志》

2025

N-嘧啶三氟乙基硫醚/亚砜苯胺类化合物的设计、合成与杀螨活性

王佳鑫，蔡胜梅，田平义，包如胜，刘祈星，周海峰

《农药》

DOI

2025

Solvent-Controlled Ring-Opening Halogenation and Halosulfonation of Alkynyl Sulfonium Salts with Alkali Halides.

Li Yang, Qian-Zhi Yang, Jia Shu, Yun Liu, Yuan-Xin Jin, Qixing Liu, Long-Yong Xie

Journal of Organic Chemistry

DOI

2025

Stereoselective Nickel-Catalyzed Iterative 1,2-Reduction of Trisubstituted Enones to Cycloalkanols Bearing Two Contiguous Stereocenters.

Yue Liu, Chao Yang, Linhong Zuo, Qixing Liu, Xu-Meng Zhang, Cheng Hou, Cong-Cong Yin, Hai-Feng Zhou

Organic Letters

DOI

2024

新型含丁烯酸内酯基三氟乙基硫醚(亚砜)类化合物的设计、合成与杀螨活性

罗时燕，陈锦彪，林健，田平义，刘祈星，周海峰

《农药学学报》

DOI

2024

机械力促进的硫醚选择性氧化制备亚砜/砜

王金龙，范吉霞，刘祈星，周海峰

《精细化工》

2024

含咪唑烷酮(吡咯甲酰胺)结构的三氟乙基硫醚(亚砜)类化合物的设计、合成及杀螨活性

陈锦彪，罗时燕，田平义，林健，刘祈星，周海峰

《农药》

2024

Water-mediated one-pot multi-step synthesis of chiral 1,3-diarylpropan-1-ols by asymmetric hydrofunctionalisation of simple alkynes

Pinke Yu, Qixing Liu, Linhong Zuo, Xu-Meng Zhang, Cong-Cong Yin, Hai-Feng Zhou

Green Chemistry

DOI

2024

Rhodium-Catalyzed Asymmetric Transfer Hydrogenation of Aryl Ketones Involving Free Phenolic Hydroxyl Group(s).

Kedi Chang, Ruilong Chou, Pinke Yu, Linhong Zuo, Qixing Liu, Xu-Mu Zhang, Cong-Cong Yin, Hai-Feng Zhou

Chemistry

DOI

2024

Iridium-Catalyzed Chemo- and Enantioselective Hydrogenation of Cycloalkenones to Access Chiral Cycloallylalcohols.

Kedi Chang, Li Yang, Yue Liu, Jinghao Cao, Linhong Zuo, Qixing Liu, Xu-Meng Zhang, Cong-Cong Yin, Hai-Feng Zhou

Organic Letters

DOI

2023

Synthesis of chiral β‐hydroxy selenides by ruthenium‐catalysed transfer hydrogenation of α‐aryl selenomethyl ketones

Qixing Liu, Meng-Xia Liu, Jin-Biao Chen, Jinlong Wang, Hai-Feng Zhou

Asian Journal of Organic Chemistry

DOI

2023

Synthesis of Chiral 2‐Oxazolidinones by Ruthenium‐Catalyzed Asymmetric Transfer Hydrogenation of 2‐ Oxazolones

Pinke Yu, Danyi Chen, Yiwen Liu, Cong-Cong Yin, Qixing Liu, Hai-Feng Zhou

Advanced Synthesis & Catalysis

DOI

2023

Catalyst- and additive-free chemoselective reduction of sulfoxides into sulfides using B2(OH)4 as a deoxygenative agent

Ji-Xia Fan, Yifan Du, Rong-Rong Zhao, Qixing Liu, Hai-Feng Zhou

Tetrahedron

DOI

2022

Bis(2-methoxyethyl)ether promoted intramolecular acceptorless dehydrogenative coupling to construct structurally diverse quinazolinones by molecular oxygen

Rong-Rong Zhao, Simiaomiao Wen, Hao Fu, Meng-Xia Liu, Qixing Liu, Hai-Feng Zhou

Green Chemistry

DOI

2022

Iridium-catalyzed chemoselective transfer hydrogenation of α, β-unsaturated ketones to saturated ketones in water

Xiao-Lan Jiang, Xiao-Feng Cui, Jinxu Chen, Qixing Liu, Yong-Sheng Chen, Hai-Feng Zhou

Tetrahedron Letters

DOI

2022

One‐pot Construction of Fluorinated Chiral Alcohols via Sequential Substitution/Asymmetric Transfer Hydrogenation of α‐Bromoarylketones and Fluoroalcohols

Rongrong Zhao, Qiaoyuan Wei, Yuxing Huang, Qing-Yue Qu, Qixing Liu, Hai-Feng Zhou

Advanced Synthesis & Catalysis

DOI

2021

氯巴占合成工艺改进

彭琛琛，张志东，刘祈星，廖宗权，周海峰

《中国医药工业杂志》

DOI

2021

Asymmetric Stepwise Reductive Amination of Aryl N ‐Heteroaryl Ketones with Benzyl Amines via Iridium Catalysis

Bing-Qin Yang, Hao Fu, Jing Yuan, Simiaomiao Wen, Chunqin Wang, Qixing Liu, Hai-Feng Zhou

Asian Journal of Organic Chemistry

DOI

2021

Ruthenium-catalysed synthesis of chiral exocyclic allylic alcohols via chemoselective transfer hydrogenation of 2-arylidene cycloalkanones

Kaili Zhang, Qixing Liu, Renke He, Danyi Chen, Zhang-Shuang Deng, N. Huang, Hai-Feng Zhou

DOI

2021

Poly(ethylene glycol) dimethyl ether mediated oxidative scission of aromatic olefins to carbonyl compounds by molecular oxygen

Tao Yu, Mingqing Guo, Simiaomiao Wen, Rong-Rong Zhao, Jinlong Wang, Yan-Li Sun, Qixing Liu, Hai-Feng Zhou

RSC Advances

DOI

2021

Access to 2‐Arylquinazolin‐4(3H)‐ones through Intramolecular Oxidative C(sp3)–H/N–H Cross‐Coupling Mediated by I2/DMSO

Simiaomiao Wen, Yi-fan Du, Yiwen Liu, X. Cui, Qixing Liu, Hai-Feng Zhou

Annalen der Pharmacie

DOI

2020

二卤海因参与的(取代苯基)-(吡啶-2-基)-甲酮类化合物的卤化反应

卢大顺，田菊燕，张福梅，陈瑛，张银，刘祈星，周海峰

《精细化工》

2020

钌催化的手性苯基/苯并噻唑甲醇的转移氢化合成

陈淡宜，张福梅，何丹，张紫媚，钟芬，文思妙妙，刘祈星，周海峰

《高等学校化学学报》

2020

Synthesis of Chiral Phenylbenzothiazole Methanol via Transfer Hydrogenation Catalyzed by Ruthenium Complexes

Danyi Chen, Fu-Yao Zhang, Dan He, Zi-Mei Zhang, Feng Zhong, Simiaomiao Wen, Qixing Liu, Hai-Feng Zhou

DOI

2020

Metal-free one-pot synthesis of N-arylsulfonamides from nitroarenes and sodium sulfinates in an aqueous medium

Xiao-Lan Jiang, Kaili Zhang, Rong-Rong Zhao, Di-Xiang Bai, Jinlong Wang, Binbin Li, Qixing Liu, Hai-Feng Zhou

DOI

2020

Redox-driven deracemization of secondary alcohols by sequential ether/O2-mediated oxidation and Ru-catalyzed asymmetric reduction

Bing-Qin Yang, Peng Cui, Yong-Sheng Chen, Qixing Liu, Hai-Feng Zhou

DOI

2019

Enantioselective Synthesis of 2‐Hydroxyalkyl Diarylphosphinates by Ruthenium‐Catalyzed Asymmetric Transfer Hydrogenation

Kaili Zhang, Yuping Yang, Huan Liu, Qixing Liu, Jinliang Lv, Hai-Feng Zhou

Advanced Synthesis and Catalysis

DOI

2019

Metal‐Free One‐Pot Synthesis of Sulfonamides from Nitroarenes and Arylsulfonyl Chlorides in Water

Kaili Zhang, Yin Zhang, Qixing Liu, Dan He, Juyan Tian, Hai-Feng Zhou

ChemistrySelect

DOI

2019

Copper-Catalyzed One-Pot Synthesis of 2,3-Dihydroquinazolin-4(1H)-ones from 2-Nitrobenzonitriles and Carbonyl Compounds Mediated by Diboronic Acid in Methanol–Water

Qixing Liu, Yuebo Sui, Yin Zhang, Kaili Zhang, Yong-Sheng Chen, Hai-Feng Zhou

Synlett : Accounts and Rapid Communications in Synthetic Organic Chemistry

DOI

2019

Metal-free one-pot three-step process for the direct conversion of aryl alkynes into secondary amines with TfOH/B2(OH)4

Yong-Sheng Chen, Sen-Sheng Liu, Peng Cui, Yin Zhang, Qixing Liu, Hai-Feng Zhou

Tetrahedron Letters

DOI

2019

Asymmetric transfer hydrogenation of cycloalkyl vinyl ketones to allylic alcohols catalyzed by ruthenium amido complexes.

Sen-Sheng Liu, Peng Cui, Juan-Juan Wang, Hai-Feng Zhou, Qixing Liu, Jinliang Lv

Organic and biomolecular chemistry

DOI

2019

One-pot synthesis of chiral β-hydroxysulfones from alkynes via aerobic oxysulfonylation and asymmetric reduction in MeOH/H2O

Peng Cui, Qixing Liu, Juan Wang, Huan Liu, Hai-Feng Zhou

Green Chemistry

DOI

2018

2-(4-芳氧苯氧基)丙酸衍生物的合成及除草活性

王春琴，刘祈星

《精细化工》

2018

Transformation of Alkynes into Chiral Alcohols via TfOH-Catalyzed Hydration and Ru-Catalyzed Tandem Asymmetric Hydrogenation.

Sen-Sheng Liu, Huan Liu, Hai-Feng Zhou, Qixing Liu, Jinliang Lv

Organic Letters

DOI

2018

Cu-catalyzed reduction of azaarenes and nitroaromatics with diboronic acid as reductant

Dan-Wei Pi, Hai-Feng Zhou, Yanmei Zhou, Qixing Liu, Renke He, G. Shen, Y. Uozumi

DOI

2018

Iridium-Catalyzed Highly Enantioselective Transfer Hydrogenation of Aryl N-Heteroaryl Ketones with N-Oxide as a Removable ortho-Substituent.

Qixing Liu, Chunqin Wang, Hai-Feng Zhou, Bai-Gui Wang, Jinliang Lv, Lu Cao, Yigang Fu

Organic Letters

DOI

2018

Silver-Mediated 2-Arylation/Alkylation/Acylation of Benzothiazoles with Aldehydes in Water

Hai-Feng Zhou, Qixing Liu, Min Hua, Chunqin Wang, Danyi Chen, Hao Fu

DOI

2018

One-pot synthesis of chiral alcohols from alkynes by CF3SO3H/ruthenium tandem catalysis

Huan Liu, Sen-Sheng Liu, Hai-Feng Zhou, Qixing Liu, Chunqin Wang

RSC Advances

DOI

2018

Metal-free Reduction of Nitro Aromatics to Amines with B2(OH)4/H2O

Hai-Feng Zhou, Y. Uozumi, Danyi Chen, Yanmei Zhou, Sen-Sheng Liu, Qixing Liu, Kaili Zhang

Synlett : Accounts and Rapid Communications in Synthetic Organic Chemistry

DOI

2017

Bifunctional Oxo-Tethered Ruthenium Complex Catalyzed Asymmetric Transfer Hydrogenation of Aryl N-Heteroaryl Ketones.

Bai-Gui Wang, Hai-Feng Zhou, Guo-Ren Lu, Qixing Liu, Xiao-Lan Jiang

Organic Letters

DOI

2017

A kind of method of asymmetric synthesis of Claritin carbinoxamine

Hai-Feng Zhou, Bai-Gui Wang, Qixing Liu, Xiao-Lan Jiang

2016

N-吡啶基-2-(4-芳氧苯氧基)丙酰胺的合成及抗肿瘤活性

刘祈星，柳爱平，黄明智

《精细化工》

2016

N-氮杂环甲基芳氧苯氧丙酰胺衍生物的抗肿瘤活性

刘祈星，柳爱平，黄明智

《三峡大学学报(自然科学版)》

2016

FeCl3‐Catalyzed Tandem Condensation/Intramolecular Nucleophilic Addition/C—C Bond Cleavage: A Concise Synthesis of 2‐Substitued Quinazolinones from 2‐Aminobenzamides and 1,3‐Diketones in Aqueous Media.

G. Shen, Hai-Feng Zhou, Yuebo Sui, Qixing Liu, K. Zou

DOI

2016

Asymmetric Synthesis of 3,4‐Dihydro‐2H‐1,2,4‐benzothiadiazine‐1,1‐dioxides Catalyzed by Scandium(III)‐inda‐Pybox.

Peng Du, Hai-Feng Zhou, Yuebo Sui, Qixing Liu, K. Zou

DOI

2015

3,4-二甲氧基苯甲酸乙酯的合成及晶体结构分析

范於菟，徐金林，武祥龙，刘祈星，王慧

《化学与生物工程》

2015

2-(4-芳氧苯氧基)丙酸类化合物的研究进展

刘祈星，柳爱平，胡艾希，黄明智，欧晓明，周海峰

《农药》

2014

N-杂环甲基2-(4-杂芳氧基苯氧基)丙酰胺的合成及除草活性

Qixing Liu, Ai-Xi Hu, Xiao-Guang Wang, Man-Xiang Lei, Xiao-Ming Ou, Ye-Guo Ren, Lu Huang, Ai-Ping Liu

DOI

2014

N -氮杂环甲氧基- O -（4-芳氧基苯基）乳酸酰胺的合成与除草活性

Qixing Liu, Ming-Zhi Huang, Ai-Ping Liu, Siqiao Nie, Man-Xiang Lei, Ye-Guo Ren, Huiping Pei, Li-Ying He, Li Hu, Ai-Xi Hu

DOI

2014

2-(4-芳氧苯氧基)丙酰胺的合成与生物活性

刘祈星

《湖南大学》

2012

N-烷氧基邻氨基苯甲酰胺衍生物的合成与生物活性

毛冠群，尹笃林，柳爱平，刘兴平，裴晖，左金江，刘祈星，孙炯，王晓光

《精细化工中间体》

2011

6-三氟甲基脲嘧啶衍生物的合成与除草生物活性

刘民华，毛冠群，左文清，唐明，韦天龙，刘祈星，吴道新，柳爱平

《精细化工中间体》

2011

芳氧苯氧羧酸除草剂HNPC-A8169的创制研究

黄路，何海军，刘祈星，雷满香，余淑英，任叶果，欧晓明，黄明智，柳爱平

《精细化工中间体》

精选作品

期刊论文

基于CVL-231的环丁胺类M4正向变构调节剂的设计、合成与活性

新型N-2,3-二氟苯基环丁胺类M4 AChR正向变构调节剂的设计、合成与活性

新型噻唑烷酮三氟乙基亚砜类化合物的设计、合成及杀螨活性

Mechanochemical NH 4 Cl-mediated hydrogen-bonding network reconstruction of HFIP: enabling yne-allylic substitutions

Nickel-Catalyzed Asymmetric Hydrogenation of All-Carbon Tetrasubstituted Alkenes Enabled by van der Waals Interactions.

盐酸曲美他嗪的合成工艺改进

含螺噻唑烷酮的三氟乙基硫醚类化合物的合成与杀螨活性

利格列汀原料药有关物质的合成

N-嘧啶三氟乙基硫醚/亚砜苯胺类化合物的设计、合成与杀螨活性

Solvent-Controlled Ring-Opening Halogenation and Halosulfonation of Alkynyl Sulfonium Salts with Alkali Halides.

Stereoselective Nickel-Catalyzed Iterative 1,2-Reduction of Trisubstituted Enones to Cycloalkanols Bearing Two Contiguous Stereocenters.

新型含丁烯酸内酯基三氟乙基硫醚(亚砜)类化合物的设计、合成与杀螨活性

机械力促进的硫醚选择性氧化制备亚砜/砜

含咪唑烷酮(吡咯甲酰胺)结构的三氟乙基硫醚(亚砜)类化合物的设计、合成及杀螨活性

Water-mediated one-pot multi-step synthesis of chiral 1,3-diarylpropan-1-ols by asymmetric hydrofunctionalisation of simple alkynes

Rhodium-Catalyzed Asymmetric Transfer Hydrogenation of Aryl Ketones Involving Free Phenolic Hydroxyl Group(s).

Iridium-Catalyzed Chemo- and Enantioselective Hydrogenation of Cycloalkenones to Access Chiral Cycloallylalcohols.

Synthesis of chiral β‐hydroxy selenides by ruthenium‐catalysed transfer hydrogenation of α‐aryl selenomethyl ketones

Synthesis of Chiral 2‐Oxazolidinones by Ruthenium‐Catalyzed Asymmetric Transfer Hydrogenation of 2‐ Oxazolones

Catalyst- and additive-free chemoselective reduction of sulfoxides into sulfides using B2(OH)4 as a deoxygenative agent

Bis(2-methoxyethyl)ether promoted intramolecular acceptorless dehydrogenative coupling to construct structurally diverse quinazolinones by molecular oxygen

Iridium-catalyzed chemoselective transfer hydrogenation of α, β-unsaturated ketones to saturated ketones in water

One‐pot Construction of Fluorinated Chiral Alcohols via Sequential Substitution/Asymmetric Transfer Hydrogenation of α‐Bromoarylketones and Fluoroalcohols

氯巴占合成工艺改进

Asymmetric Stepwise Reductive Amination of Aryl N ‐Heteroaryl Ketones with Benzyl Amines via Iridium Catalysis

Ruthenium-catalysed synthesis of chiral exocyclic allylic alcohols via chemoselective transfer hydrogenation of 2-arylidene cycloalkanones

Poly(ethylene glycol) dimethyl ether mediated oxidative scission of aromatic olefins to carbonyl compounds by molecular oxygen

Access to 2‐Arylquinazolin‐4(3H)‐ones through Intramolecular Oxidative C(sp3)–H/N–H Cross‐Coupling Mediated by I2/DMSO

二卤海因参与的(取代苯基)-(吡啶-2-基)-甲酮类化合物的卤化反应

钌催化的手性苯基/苯并噻唑甲醇的转移氢化合成

Synthesis of Chiral Phenylbenzothiazole Methanol via Transfer Hydrogenation Catalyzed by Ruthenium Complexes

Metal-free one-pot synthesis of N-arylsulfonamides from nitroarenes and sodium sulfinates in an aqueous medium

Redox-driven deracemization of secondary alcohols by sequential ether/O2-mediated oxidation and Ru-catalyzed asymmetric reduction

Enantioselective Synthesis of 2‐Hydroxyalkyl Diarylphosphinates by Ruthenium‐Catalyzed Asymmetric Transfer Hydrogenation

Metal‐Free One‐Pot Synthesis of Sulfonamides from Nitroarenes and Arylsulfonyl Chlorides in Water

Copper-Catalyzed One-Pot Synthesis of 2,3-Dihydroquinazolin-4(1H)-ones from 2-Nitrobenzonitriles and Carbonyl Compounds Mediated by Diboronic Acid in Methanol–Water

Metal-free one-pot three-step process for the direct conversion of aryl alkynes into secondary amines with TfOH/B2(OH)4

Asymmetric transfer hydrogenation of cycloalkyl vinyl ketones to allylic alcohols catalyzed by ruthenium amido complexes.

One-pot synthesis of chiral β-hydroxysulfones from alkynes via aerobic oxysulfonylation and asymmetric reduction in MeOH/H2O

2-(4-芳氧苯氧基)丙酸衍生物的合成及除草活性

Transformation of Alkynes into Chiral Alcohols via TfOH-Catalyzed Hydration and Ru-Catalyzed Tandem Asymmetric Hydrogenation.

Cu-catalyzed reduction of azaarenes and nitroaromatics with diboronic acid as reductant

Iridium-Catalyzed Highly Enantioselective Transfer Hydrogenation of Aryl N-Heteroaryl Ketones with N-Oxide as a Removable ortho-Substituent.

Silver-Mediated 2-Arylation/Alkylation/Acylation of Benzothiazoles with Aldehydes in Water

One-pot synthesis of chiral alcohols from alkynes by CF3SO3H/ruthenium tandem catalysis

Metal-free Reduction of Nitro Aromatics to Amines with B2(OH)4/H2O

Bifunctional Oxo-Tethered Ruthenium Complex Catalyzed Asymmetric Transfer Hydrogenation of Aryl N-Heteroaryl Ketones.

A kind of method of asymmetric synthesis of Claritin carbinoxamine

N-吡啶基-2-(4-芳氧苯氧基)丙酰胺的合成及抗肿瘤活性

N-氮杂环甲基芳氧苯氧丙酰胺衍生物的抗肿瘤活性

FeCl3‐Catalyzed Tandem Condensation/Intramolecular Nucleophilic Addition/C—C Bond Cleavage: A Concise Synthesis of 2‐Substitued Quinazolinones from 2‐Aminobenzamides and 1,3‐Diketones in Aqueous Media.

Asymmetric Synthesis of 3,4‐Dihydro‐2H‐1,2,4‐benzothiadiazine‐1,1‐dioxides Catalyzed by Scandium(III)‐inda‐Pybox.

3,4-二甲氧基苯甲酸乙酯的合成及晶体结构分析

2-(4-芳氧苯氧基)丙酸类化合物的研究进展

N-杂环甲基2-(4-杂芳氧基苯氧基)丙酰胺的合成及除草活性

N -氮杂环甲氧基- O -（4-芳氧基苯基）乳酸酰胺的合成与除草活性

2-(4-芳氧苯氧基)丙酰胺的合成与生物活性

N-烷氧基邻氨基苯甲酰胺衍生物的合成与生物活性

6-三氟甲基脲嘧啶衍生物的合成与除草生物活性

芳氧苯氧羧酸除草剂HNPC-A8169的创制研究

会议论文

二硼试剂参与的硝基还原及串联反应研究

N-氧化物为瞬态邻位取代基策略:手性二胺铱络合物催化的芳基-氮杂芳基甲酮不对称转移氢化

研究方向