冯煌迪｜上海工程技术大学｜学者主页

2026

Cycloaddition Enables Ring Opening of N -Propargyl Oxazolidines: Access to N -Benzyl-2,3-diphenylpyrroles via Both C–O and C–C Bond Cleavage

Siyan Qiu, Ya Pan, Tingyu Zhang, Jinglong Kong, Junhai Huang, Huangdi Feng

The Journal of Organic Chemistry

DOI

2026

Streamlined access to diversified 3-aminothiophene building blocks via a neat tandem reaction sequence

Peng Li, Ziqi Yi, Chuang Liu, Jingxuan Nie, Jiaxin Huang, Huangdi Feng, Junhai Huang

Tetrahedron

DOI

2026

Ortho ‐Alkynyl Quinone Methides as Privileged Intermediates in Synthesis of Polycyclic Frameworks: A Short Review

Shuangshuang Liu, Wenjing Hou, Liliang Huang, Huangdi Feng

The Chemical Record

DOI

2026

Deoxygenative C(sp 3 )–S Cross-Coupling of Alcohols and Sulfenamides

Wentong Liu, Yifan Liu, Liliang Huang, Junhai Huang, Huangdi Feng

The Journal of Organic Chemistry

DOI

2026

Ring-Restructuring of gem-Difluorocyclopropanes: Diverse Access to Four- to Nine-Membered Ring Skeletons

Yan Sun, Chao Yang, Liliang Huang, Huangdi Feng

Pharmaceutical Fronts

DOI

2026

Facile construction of bis-spiro-enol oxazolidines via a modular tandem strategy

Rongkang Zhang, Yong Qian, Liliang Huang, Junhai Huang, Huangdi Feng

Tetrahedron Letters

DOI

2025

Regioselective Difunctionalization of gem -Difluorocyclopropanes via Palladium-Catalyzed Defluorinative Coupling

Chao Yang, Liliang Huang, Youcan Zhang, Yong Qian, Zhenjie Wang, Huangdi Feng

The Journal of Organic Chemistry

DOI

2025

One-Pot Assembly of 2-Pyrones through Copper-Catalyzed Cyclization of Propargylamines with Malonates

Junwei Li, Shuangshuang Liu, Liliang Huang, Junhai Huang, Huangdi Feng

Precision Chemistry

DOI

2025

Streamlined Deamination of Diverse Primary Amines Enabled by Anomeric Amide

Ya Pan, Wentong Liu, Liliang Huang, Junhai Huang, Huangdi Feng

Chinese Journal of Chemistry

DOI

2025

S-Benzylation of Sulfenamides with Tertiary Amine Using Methyl Propiolate as a Bifunctional Additive

Wentong Liu, Siyan Qiu, Ruiyang Jin, Liliang Huang, Junhai Huang, Huangdi Feng

The Journal of Organic Chemistry

DOI

2025

Approved alkyne-containing drugs: A review of their pharmacokinetic properties and therapeutic applications

Jing Wang, Aiguo Gu, Huangdi Feng, Chuang Liu, Peng Li, Junhai Huang

European Journal of Medicinal Chemistry

DOI

2025

Access to 1,6-Enynes via Cadmium-Catalyzed Domino A 3 -Coupling/Dealkylative A 3 -Coupling

Tiantian Zhang, Ming He, Siyan Qiu, Liliang Huang, Junhai Huang, Huangdi Feng

Organic Letters

DOI

2025

Alkyne‐Dependent Synthesis of Pyrrolines and Propargylamines through Metal‐Free Decarboxylation

Ziqi Yi, Peng Li, Shuailin Fan, Huangdi Feng, Junhai Huang

European Journal of Organic Chemistry

DOI

2025

Copper(I)-Catalyzed Synthesis of 1-Amino-1,3-diene Derivatives through a Formal 1,3-Amino Migration Process

Junwei Li, Shuangshuang Liu, Tiantian Zhang, Liliang Huang, Huangdi Feng

Organic Letters

DOI

2025

Synthesis of indolizines via Pd-catalyzed selective ring recasting of oxazolidines with deesterification of methyl acrylates

Ya Pan, Xianjun Xu, Junwei Li, Luosang Cuomu, Erik V. Van der Eycken, Huangdi Feng

Sustainable Chemistry and Pharmacy

DOI

2025

Base-promoted efficient transformation of aryl methylene bromides and DMSO to vinyl sulfoxides

Aiguo Gu, Xiaofan Shi, Junhai Huang, Rongkang Zhang, Liliang Huang, Huangdi Feng

Tetrahedron Letters

DOI

2025

Synthesis of Tetrasubstituted Pyrroles via DBU-Mediated Cyclization of Unactivated Propargyl Tertiary Amines

Pengyu Zhou, Tiantian Zhang, Qing Lu, Yujuan Xie, Liliang Huang, Huangdi Feng

The Journal of Organic Chemistry

DOI

2025

Assembly of Diverse Allenes via Activator-Free Palladium-Catalyzed Regioselective γ-Arylation of Propargylamines with Boronic Acids

Yan Lin Sun, Ya Pan, Tao Zhao, Junwei Li, Aiguo Gu, Junhai Huang, Huangdi Feng

The Journal of Organic Chemistry

DOI

2025

Copper-Catalyzed Four-Component A3-Based Cascade Reaction: Facile Synthesis of 3-Oxetanone-Derived Spirocycles

Rongkang Zhang, Liliang Huang, Aiguo Gu, Huangdi Feng

Chemistry

DOI

2025

A Cu/Cd-cocatalysed cascade reaction for constructing nitrogen-tethered 1,6-enynes enabled by 1,5-hydride transfer

Tiantian Zhang, Hexiang Wang, Liliang Huang, Junhai Huang, Huangdi Feng

Organic Chemistry Frontiers

DOI

2024

Asymmetric synthesis of atropisomers featuring cyclobutane boronic esters facilitated by ring-strained B-ate complexes

Yu-Wen Sun, Jia-Hui Zhao, Xinyu Yan, Chong‐Lei Ji, Huangdi Feng, De‐Wei Gao

Nature Communications

DOI

2024

Efficient synthesis of trisubstituted allenes via palladium-catalysed deaminative coupling of tertiary propargylamines with arylsiloxanes

Mingjie Liao, Ziqi Yi, Qingqing You, Chuang Liu, Huangdi Feng, Junhai Huang

Organic Chemistry Frontiers

DOI

2024

Advancements in Desilylation Reactions for the Synthesis of Valuable Organic Molecules

Chuang Liu, Le Zhang, Qingqing You, Huangdi Feng, Junhai Huang

The Chemical Record

DOI

2024

Facile synthesis of vinyl sulfoxides via external oxidant-free oxidative condensation of phenylglycinols with DMSO

Xiaofan Shi, Rongkang Zhang, Chuang Liu, Zhicheng Zuo, Huangdi Feng

Tetrahedron Letters

DOI

2024

Catalytic Selective Functionalization of Poly(organoborons)†

Jiahui Zhao, Ang Chen, Xi‐Zhang Zou, Chong‐Lei Ji, Huangdi Feng, De‐Wei Gao

Chinese Journal of Chemistry

DOI

2024

A novel propiolate-enabled deaminative hiyama coupling of aryl silanes and propargylamines

Qingqing You, Chuang Liu, Mingjie Liao, Huangdi Feng, Junhai Huang

Molecular Catalysis

DOI

2024

Metal- and oxidant-free skeletal reorganizing of oxazolidines to access N-Vinylpyrroles

Ruidan Shi, Xianjun Xu, Ling Zhong, Leilei Cao, Ya Pan, Junhai Huang, Huangdi Feng

Sustainable Chemistry and Pharmacy

DOI

2024

Organocatalytic Deoxygenative [3+2] Cycloaddition of N-Hydroxyamides with Alkynes to Access Isoxazoles

Haixiang Wang, Yan Lin Sun, Wentong Liu, Liliang Huang, Huangdi Feng

Organic Letters

DOI

2024

Precision Propargylic Substitution Reaction: Pd-Catalyzed Suzuki–Miyaura Coupling of Nonactivated Propargylamines with Boronic Acids

Yan Lin Sun, Tao Zhao, Haixiang Wang, Ya Pan, Liliang Huang, Huangdi Feng

The Journal of Organic Chemistry

DOI

2024

Palladium-Catalyzed Regioselective Monofluoroallylation of Indoles with gem -Difluorocyclopropanes

Zhenjie Wang, Chuang Liu, Junhai Huang, Liliang Huang, Huangdi Feng

Organic Letters

DOI

2024

Skeletal Editing of Isatins for Heterocycle Molecular Diversity

Tiantian Zhang, Huangdi Feng

The Chemical Record

DOI

2024

Ring expansion strategy to access functionalized 2-oxazolines (microreview)

L.‐G. LIU, Wentong Liu, Huangdi Feng

Chemistry of Heterocyclic Compounds

DOI

2024

Cover Picture: Skeletal Editing of Isatins for Heterocycle Molecular Diversity (Chem. Rec. 6/2024)

Tiantian Zhang, Huangdi Feng

The Chemical Record

DOI

2024

Microwave-assisted palladium-catalyzed conjugate addition of arylsilanes to alkynes

Mingjie Liao, Chuang Liu, Huangdi Feng, Qingqing You, Junhai Huang

Molecular Catalysis

DOI

2024

Transition-metal-free Csp–Csp doubly decarboxylative coupling of amino acids and propiolic acids

Junduo Hu, L.‐G. LIU, Haixiang Wang, Liliang Huang, Huanmei Gao, Huangdi Feng

Sustainable Chemistry and Pharmacy

DOI

2024

Facile synthesis of propargylamines by metal-free doubly decarboxylative coupling

Junduo Hu, Xiaofan Shi, Liliang Huang, Rongkang Zhang, Huangdi Feng

RSC Sustainability

DOI

2023

Synthesis of oxazolines through a Pd-catalyzed alkyne-enabled C N activation of oxazolidines

Ling Zhong, Ruidan Shi, Liliang Huang, Junhai Huang, Huangdi Feng

Tetrahedron Letters

DOI

2023

Pictet–Spengler-Based Multicomponent Domino Reactions to Construct Polyheterocycles

Junduo Hu, Liliang Huang, Huangdi Feng

Pharmaceutical Fronts

DOI

2023

CuS Morphology Control for Enhanced Catalytic Performance in A 3 Coupling Reaction

Sainan Cao, Yongqi Pan, Huangdi Feng, Jingxia Yang

ChemistrySelect

DOI

2023

Application of Metal‐Free Dearomatization Reaction as a Sustainable Strategy to Direct Access Complex Cyclic Compounds

Xianjun Xu, Ling Zhong, Huangdi Feng, Erik V. Van der Eycken

The Chemical Record

DOI

2023

Metal-catalyst- and fluoride-free oxidative desilylation of arylsilanes and its application

Qingqing You, Liliang Huang, Mingjie Liao, Yuchen Meng, Huangdi Feng, Junhai Huang

Sustainable Chemistry and Pharmacy

DOI

2022

苯并噁唑类化合物的制备综合实验设计

黄立梁，冯煌迪

《广东化工》

2022

Amine-catalyzed metal-free deamination of propargylamines with water toward chalcones

Pengyu Zhou, Liliang Huang, Yujuan Xie, Gaoxiang Ma, Huangdi Feng

Molecular Catalysis

DOI

2022

Hollow CuO–CeO2 Nanospheres for an Effectively Catalytic Annulation/A3-Coupling Reaction Sequence

Sainan Cao, Bingjie Zou, Jingxia Yang, Jinjie Wang, Huangdi Feng

ACS Applied Nano Materials

DOI

2022

Vinyl fluorosulfonamide: a practical vinyl electrophilic reagent for mild and efficient synthesis of ketones under catalyst- and additive-free conditions

Bin Qing, Xueying Bai, Liliang Huang, Jiahui Zhao, Pengyu Zhou, Huangdi Feng

Phosphorus, sulfur, and silicon and the related elements

DOI

2022

Synthesis of pyrroles from propargylamines and their derivatives: an update (microreview)

Jingyi Gong, Huangdi Feng

Chemistry of Heterocyclic Compounds

DOI

2022

Selectivity Controlled Hydroamination of Alkynes to Sulfonyl Fluoride Hubs: Development and Application

Xueying Bai, Liliang Huang, Pengyu Zhou, Hui Xi, Junduo Hu, Zhicheng Zuo, Huangdi Feng

The Journal of Organic Chemistry

DOI

2022

Direct Access to 4-Substituted Isoquinolones via a Sequential Pd-Catalyzed Cyclization/Base-Promoted Aromatization/Ring-Opening of N-Propargyl-1,3-oxazolidines

Xianjun Xu, Liangliang Song, Huangdi Feng, Erik V. Van der Eycken

Molecular Catalysis

DOI

2022

Accessing N‐Propargyl Amino Alcohols through Cu(I)‐Catalyzed A 3 ‐Coupling/Annulation and Bi(III)‐Promoted Ring‐Opening

Leilei Cao, Pengyu Zhou, Junduo Hu, Liliang Huang, Huangdi Feng

ChemistrySelect

DOI

2022

Pd-Catalyzed Ring Restructuring of Oxazolidines with Alkenes Leading to Fused Polycyclic Indolizines

Xianjun Xu, Huangdi Feng, Xiaoyong Zhang, Liangliang Song, Luc Van Meervelt, Johan Van der Eycken, Jeremy Noel Harvey, Erik V. Van der Eycken

Organic Letters

DOI

2022

A highly efficient metal-free hydrocarbonylation of alkynes with propargylamines and water

Yujuan Xie, Liliang Huang, Yayu Qi, Junduo Hu, Liangliang Song, Huangdi Feng

Green Chemistry

DOI

2022

Microwave-assisted decarboxylative reactions: advanced strategies for sustainable organic synthesis

Qingqing You, Mingjie Liao, Huangdi Feng, Junhai Huang

Organic & Biomolecular Chemistry

DOI

2022

Synthesis of N -alkenylisoquinolinones via palladium-catalyzed cyclization/C 4 –O bond cleavage of oxazolidines

Xianjun Xu, Liliang Huang, Eva Smits, Ling Zhong, Huangdi Feng, Erik V. Van der Eycken

New Journal of Chemistry

DOI

2021

aza-Morita-Baylis-Hillman反应二次串联构建氨基衍生的1,6-二烯化合物

彭福涛，黄立梁，黄军海，冯煌迪

《有机化学》

2021

Synthesis of nitrogen-tethered 1,6-enynes through CuI/TFA catalysis

Leilei Cao, Liliang Huang, Xianjun Xu, Erik V. Van der Eycken, Huangdi Feng

Organic Chemistry Frontiers

DOI

2021

Chemodivergent Synthesis of Oxazolidin-2-ones via Cu-Catalyzed Carboxyl Transfer Annulation of Propiolic Acids with Amines

Yujuan Xie, Huangdi Feng, Yayu Qi, Junhai Huang, Liliang Huang

The Journal of Organic Chemistry

DOI

2021

Recent Advances in the Synthesis and Ring‐Opening Transformations of 2‐Oxazolidinones

Feixiang Sun, Erik V. Van der Eycken, Huangdi Feng

Advanced Synthesis & Catalysis

DOI

2021

Catalyst‐Free Hydrogen Proton Transfer Reduction of Nitrobenzamides to Aminobenzamides with iPrOH/KOH System

Xueying Bai, Liliang Huang, Bin Qing, Zhicheng Zuo, Huangdi Feng

Asian Journal of Organic Chemistry

DOI

2021

Microwave-Assisted Palladium-Catalyzed Reductive Cyclization/Ring-Opening/Aromatization Cascade of Oxazolidines to Isoquinolines

Xianjun Xu, Huangdi Feng, Erik V. Van der Eycken

Organic Letters

DOI

2021

Switchable Mono‐ and Dipropargylation of Amino Alcohols: A Unique Property of the Iodide Anion in Controlling Ring‐Opening Alkynylation

Huangdi Feng, Fang Wang, Leilei Cao, Erik V. Van der Eycken, Xiaoying Yin

European Journal of Organic Chemistry

DOI

2021

RECENT ADVANCES IN DEAROMATIZATION OF BENZAZOLES, PURINES, AND CAFFEINE

Liliang Huang, Huangdi Feng

Chemistry of Heterocyclic Compounds

DOI

2021

Recent advances in dearomatization of benzazoles, purines, and caffeine (microreview)

Liliang Huang, Huangdi Feng

Chemistry of Heterocyclic Compounds

DOI

2021

Microwave-Assisted Cu(I)-Catalyzed Synthesis of Unsymmetrical 1,4-Diamino-2-butynes via Cross-A3-Coupling/Decarboxylative A3-Coupling

Xianjun Xu, Huangdi Feng, Erik V. Van der Eycken

The Journal of Organic Chemistry

DOI

2021

Glyoxylic Acid: A Carboxyl Group‐Assisted Metal‐Free Decarboxylative Reaction Toward Propargylamines

Liliang Huang, Yujuan Xie, Panyuan Ge, Junhai Huang, Huangdi Feng

European Journal of Organic Chemistry

DOI

2021

Cu‐Catalyzed Selective Synthesis of Propargylamines via A3‐Coupling/Aza‐Michael Addition Sequence: Amine Loading Controls the Selectivity

Huangdi Feng, Futao Peng, Hui Xi, Ling Zhong, Liliang Huang

Asian Journal of Organic Chemistry

DOI

2021

Modular Synthesis of Unsymmetrical 1,4‐Diamino‐2‐butynes by Cu–Catalyzed Sequential Decarboxylative A3‐Coupling/Petasis Reaction/A3‐Coupling

Shuangyuan Zhu, Huangdi Feng, Shengyun Hu, Tingting Guo, Ming Li, Shaoying Tan, Liliang Huang, Junhai Huang

Asian Journal of Organic Chemistry

DOI

2021

Copper-catalyzed deaminative alkynylation of secondary amines with alkynes: selectivity switch in the synthesis of diverse propargylamines

Shengyun Hu, Huangdi Feng, Hui Xi, Yuchen Meng, Ming Li, Liliang Huang, Junhai Huang

Organic Chemistry Frontiers

DOI

2021

CF 3 SO 3 H-enabled cascade ring-opening/dearomatization of indole derivatives to polycyclic heterocycles

Zhengdong Yao, Huangdi Feng, Hui Xi, Chuanjun Xi, Weiping Liu

Organic & Biomolecular Chemistry

DOI

2020

铜(Ⅰ)催化丙炔酸、仲胺、醛和甲醛一锅法交叉偶联构建非对称1,4-二氨基丁炔

刘博瑜，徐仙君，黄立梁，冯煌迪

《有机化学》

2020

Ynoate-Initiated Selective C–N Esterification of Tertiary Amines under Transition-Metal and Oxidant-Free Conditions

Huangdi Feng, Junhai Huang, Feixiang Sun, Liliang Huang

Synlett

DOI

2020

A lysosome specific ratiometric fluorescent probe for detection of bisulfite ion based on hybrid coumarin-benzimidazolium compounds

Jiangdong Zhao, Liliang Huang, Meiling Yan, Yi Qu, Huangdi Feng, Yanhong Sun

Phosphorus, sulfur, and silicon and the related elements

DOI

2020

Lewis Acid‐Free Ynoate‐Mediated Chemoselective Reduction of Carboxylic Acids to Primary Alcohols

Feixiang Sun, Huangdi Feng, Liliang Huang, Weiping Liu

ChemistrySelect

DOI

2020

Metal‐Free Decarboxylation of α, β‐Unsaturated Carboxylic Acids for Carbon–Carbon and Carbon–Heteroatom Coupling Reactions

Xianjun Xu, Erik V. Van der Eycken, Huangdi Feng

Chinese Journal of Chemistry

DOI

2020

DOMINO DECARBOXYLATION–CO 2 FIXATION – A ROUTE TOWARD CYCLIC CARBONATES AND OXAZOLIDINONES

Huangdi Feng

Chemistry of Heterocyclic Compounds

DOI

2020

Domino Decarboxylation–CO2 Fixation – a Route toward Cyclic Carbonates and Oxazolidinones (Microreview)

Huangdi Feng

Chemistry of Heterocyclic Compounds

DOI

2020

Synthesis of functionalized oxazolidines by multicomponent reactions of 1,2-amino alcohols (microreview)

Xianjun Xu, Hua Wei, Huangdi Feng

Chemistry of Heterocyclic Compounds

DOI

2020

Metal‐Free Decarboxylative A3‐Coupling/Pictet–Spengler Cascade Accessing Polycyclic Scaffolds: Propiolic Acids Exceed Alkynes

Yingxin Hu, Yangpeng Shen, Liliang Huang, Erik V. Van der Eycken, Huangdi Feng

European Journal of Organic Chemistry

DOI

2019

1D Fe3O4@CuSiO3 composites catalyzed decarboxylative A3-coupling for propargylamine synthesis

Fang Wang, Huangdi Feng, Huiqiong Li, Teng Miao, Tiantian Cao, Min Zhang

Chinese Chemical Letters

DOI

2019

Synthesis of γ-(Arylamino)butyric Acid Derivatives via Ring-Opening Addition of Arylamines to Cyclopropane-1,1-Dicarboxylates

S. K. Li, Liliang Huang, Yandong Lv, Huangdi Feng

Russian Journal of Organic Chemistry

DOI

2019

Synthetic Access to Secondary Propargylamines via a Copper-Catalyzed Oxidative Deamination/Alkynylation Cascade

Huiqiong Li, Huangdi Feng, Jingxian Zhang, Erik V. Van der Eycken, Liliang Huang

The Journal of Organic Chemistry

DOI

2019

Carboxyl Transfer of α-Keto Acids toward Oxazolidinones via Decarboxylation/Fixation of Liberated CO2

Huiqiong Li, Huangdi Feng, Fang Wang, Liliang Huang

The Journal of Organic Chemistry

DOI

2019

Synthesis, characterization and biological activity of 1,3-diazaheteroaromatic derivatives by the ring-opening domino reaction

Shikang Li, Liliang Huang, Zhuo Chen, Jiangdong Zhao, Huangdi Feng

Journal of Molecular Structure

DOI

2019

Enol Ester Intermediate Induced Metal‐Free Oxidative Coupling of Carboxylic Acids and Arylboronic Acids

Xianjun Xu, Huangdi Feng, Huiqiong Li, Liliang Huang

European Journal of Organic Chemistry

DOI

2019

Chemo- and Diastereoselective Synthesis of N-Propargyl Oxazolidines through a Copper-Catalyzed Domino A3 Reaction

Yazhen Zhang, Liliang Huang, Xiaoyang Li, Le Wang, Huangdi Feng

The Journal of Organic Chemistry

DOI

2019

Copper‐Catalyzed Annulation/A3‐Coupling Cascade: Diastereodivergent Synthesis of Sterically Hindered Monocyclic Oxazolidines Bearing Multiple Stereocenters

Huangdi Feng, Yazhen Zhang, Zedi Zhang, Fubei Chen, Liliang Huang

European Journal of Organic Chemistry

DOI

2018

Direct Amidation of Carboxylic Acids through an Active α-Acyl Enol Ester Intermediate

Xianjun Xu, Huangdi Feng, Liliang Huang, Xiaohui Liu

The Journal of Organic Chemistry

DOI

2018

A Highly Chemoselective Synthesis of Cyclic Divalent Propargylamines by Copper‐Catalyzed Annulation/Double A3‐Couplings

Yazhen Zhang, Huangdi Feng, Xiaohui Liu, Liliang Huang

European Journal of Organic Chemistry

DOI

2018

Dual roles of ynoates: desymmetrization of dicarboxylic acids using trialkylamines as alkyl equivalents

Xianjun Xu, Liliang Huang, Xiaoying Yin, Erik V. Van der Eycken, Huangdi Feng

Organic Chemistry Frontiers

DOI

2016

Highly Selective Synergistic Copper(I/II)‐Catalyzed A3 Cross Coupling/Decarboxylative A3 Domino Reactions in Water

Huangdi Feng, Zhao Panfeng, Liliang Huang, Zhihua Sun, Min‐Chao Tong

Asian Journal of Organic Chemistry

DOI

2016

Controlling chemoselectivity in copper-catalyzed decarboxylative A 3 /A 3 cross-couplings: direct formation of unsymmetrical 1,4-diamino-2-butynes

Zhao Panfeng, Huangdi Feng, Haoran Pan, Zhihua Sun, Min‐Chao Tong

Organic Chemistry Frontiers

DOI

2015

CuI/CuBr2-catalyzed decarboxylative/A3 reaction of propiolic acids for the facile synthesis of 1,4-diheterocycle-2-butynes

Huangdi Feng, Zhao Panfeng, Zhihua Sun

Tetrahedron Letters

DOI

2015

A Metal‐Free Approach Toward Saturated N‐Propargyl Heterocycles via an Annulation/Decarboxylative Coupling Sequence

Huangdi Feng, Huihui Jia, Zhihua Sun

Advanced Synthesis & Catalysis

DOI

2015

Decarboxylative dipropargylation of primary amines with propiolic acids and formaldehyde via metal-free coupling

Huihui Jia, Huangdi Feng, Zhihua Sun

Tetrahedron

DOI

2015

Multicomponent domino reactions of hydrazinecarbodithioates: concise access to 3-substituted 5-thiol-1,3,4-thiadiazolines

Huihui Jia, Huangdi Feng, Zhihua Sun

Organic & Biomolecular Chemistry

DOI

2014

Mild and Catalyst-Free Petasis/Decarboxylative Domino Reaction: Chemoselective Synthesis of N -Benzyl Propargylamines

Huangdi Feng, Huihui Jia, Zhihua Sun

The Journal of Organic Chemistry

DOI

2014

Pd-NHC-catalyzed synthesis of diaryl ketones

Feng Gao, Huangdi Feng, Zhihua Sun

Tetrahedron Letters

DOI

2014

Nano Cu-catalyzed efficient and selective reduction of nitroarenes under combined microwave and ultrasound irradiation

Huangdi Feng, Yuan Li, Shengji Lin, Erik V. Van der Eycken, Gonghua Song

Sustainable Chemical Processes

DOI

2012

微波促进或微波-超声复合场促进多组分反应

冯煌迪

《华东理工大学》

精选作品

期刊论文

Cycloaddition Enables Ring Opening of N -Propargyl Oxazolidines: Access to N -Benzyl-2,3-diphenylpyrroles via Both C–O and C–C Bond Cleavage

Streamlined access to diversified 3-aminothiophene building blocks via a neat tandem reaction sequence

Ortho ‐Alkynyl Quinone Methides as Privileged Intermediates in Synthesis of Polycyclic Frameworks: A Short Review

Deoxygenative C(sp 3 )–S Cross-Coupling of Alcohols and Sulfenamides

Ring-Restructuring of gem-Difluorocyclopropanes: Diverse Access to Four- to Nine-Membered Ring Skeletons

Facile construction of bis-spiro-enol oxazolidines via a modular tandem strategy

Regioselective Difunctionalization of gem -Difluorocyclopropanes via Palladium-Catalyzed Defluorinative Coupling

One-Pot Assembly of 2-Pyrones through Copper-Catalyzed Cyclization of Propargylamines with Malonates

Streamlined Deamination of Diverse Primary Amines Enabled by Anomeric Amide

S-Benzylation of Sulfenamides with Tertiary Amine Using Methyl Propiolate as a Bifunctional Additive

Approved alkyne-containing drugs: A review of their pharmacokinetic properties and therapeutic applications

Access to 1,6-Enynes via Cadmium-Catalyzed Domino A 3 -Coupling/Dealkylative A 3 -Coupling

Alkyne‐Dependent Synthesis of Pyrrolines and Propargylamines through Metal‐Free Decarboxylation

Copper(I)-Catalyzed Synthesis of 1-Amino-1,3-diene Derivatives through a Formal 1,3-Amino Migration Process

Synthesis of indolizines via Pd-catalyzed selective ring recasting of oxazolidines with deesterification of methyl acrylates

Base-promoted efficient transformation of aryl methylene bromides and DMSO to vinyl sulfoxides

Synthesis of Tetrasubstituted Pyrroles via DBU-Mediated Cyclization of Unactivated Propargyl Tertiary Amines

Assembly of Diverse Allenes via Activator-Free Palladium-Catalyzed Regioselective γ-Arylation of Propargylamines with Boronic Acids

Copper-Catalyzed Four-Component A3-Based Cascade Reaction: Facile Synthesis of 3-Oxetanone-Derived Spirocycles

A Cu/Cd-cocatalysed cascade reaction for constructing nitrogen-tethered 1,6-enynes enabled by 1,5-hydride transfer

Asymmetric synthesis of atropisomers featuring cyclobutane boronic esters facilitated by ring-strained B-ate complexes

Efficient synthesis of trisubstituted allenes via palladium-catalysed deaminative coupling of tertiary propargylamines with arylsiloxanes

Advancements in Desilylation Reactions for the Synthesis of Valuable Organic Molecules

Facile synthesis of vinyl sulfoxides via external oxidant-free oxidative condensation of phenylglycinols with DMSO

Catalytic Selective Functionalization of Poly(organoborons)†

A novel propiolate-enabled deaminative hiyama coupling of aryl silanes and propargylamines

Metal- and oxidant-free skeletal reorganizing of oxazolidines to access N-Vinylpyrroles

Organocatalytic Deoxygenative [3+2] Cycloaddition of N-Hydroxyamides with Alkynes to Access Isoxazoles

Precision Propargylic Substitution Reaction: Pd-Catalyzed Suzuki–Miyaura Coupling of Nonactivated Propargylamines with Boronic Acids

Palladium-Catalyzed Regioselective Monofluoroallylation of Indoles with gem -Difluorocyclopropanes

Skeletal Editing of Isatins for Heterocycle Molecular Diversity

Ring expansion strategy to access functionalized 2-oxazolines (microreview)

Cover Picture: Skeletal Editing of Isatins for Heterocycle Molecular Diversity (Chem. Rec. 6/2024)

Microwave-assisted palladium-catalyzed conjugate addition of arylsilanes to alkynes

Transition-metal-free Csp–Csp doubly decarboxylative coupling of amino acids and propiolic acids

Facile synthesis of propargylamines by metal-free doubly decarboxylative coupling

Synthesis of oxazolines through a Pd-catalyzed alkyne-enabled C N activation of oxazolidines

Pictet–Spengler-Based Multicomponent Domino Reactions to Construct Polyheterocycles

CuS Morphology Control for Enhanced Catalytic Performance in A 3 Coupling Reaction

Application of Metal‐Free Dearomatization Reaction as a Sustainable Strategy to Direct Access Complex Cyclic Compounds

Metal-catalyst- and fluoride-free oxidative desilylation of arylsilanes and its application

苯并噁唑类化合物的制备综合实验设计

Amine-catalyzed metal-free deamination of propargylamines with water toward chalcones

Hollow CuO–CeO2 Nanospheres for an Effectively Catalytic Annulation/A3-Coupling Reaction Sequence

Vinyl fluorosulfonamide: a practical vinyl electrophilic reagent for mild and efficient synthesis of ketones under catalyst- and additive-free conditions

Synthesis of pyrroles from propargylamines and their derivatives: an update (microreview)

Selectivity Controlled Hydroamination of Alkynes to Sulfonyl Fluoride Hubs: Development and Application

Direct Access to 4-Substituted Isoquinolones via a Sequential Pd-Catalyzed Cyclization/Base-Promoted Aromatization/Ring-Opening of N-Propargyl-1,3-oxazolidines

Accessing N‐Propargyl Amino Alcohols through Cu(I)‐Catalyzed A 3 ‐Coupling/Annulation and Bi(III)‐Promoted Ring‐Opening

Pd-Catalyzed Ring Restructuring of Oxazolidines with Alkenes Leading to Fused Polycyclic Indolizines

A highly efficient metal-free hydrocarbonylation of alkynes with propargylamines and water

Microwave-assisted decarboxylative reactions: advanced strategies for sustainable organic synthesis

Synthesis of N -alkenylisoquinolinones via palladium-catalyzed cyclization/C 4 –O bond cleavage of oxazolidines

aza-Morita-Baylis-Hillman反应二次串联构建氨基衍生的1,6-二烯化合物

Synthesis of nitrogen-tethered 1,6-enynes through CuI/TFA catalysis

Chemodivergent Synthesis of Oxazolidin-2-ones via Cu-Catalyzed Carboxyl Transfer Annulation of Propiolic Acids with Amines

Recent Advances in the Synthesis and Ring‐Opening Transformations of 2‐Oxazolidinones

Catalyst‐Free Hydrogen Proton Transfer Reduction of Nitrobenzamides to Aminobenzamides with iPrOH/KOH System

Microwave-Assisted Palladium-Catalyzed Reductive Cyclization/Ring-Opening/Aromatization Cascade of Oxazolidines to Isoquinolines

Switchable Mono‐ and Dipropargylation of Amino Alcohols: A Unique Property of the Iodide Anion in Controlling Ring‐Opening Alkynylation

RECENT ADVANCES IN DEAROMATIZATION OF BENZAZOLES, PURINES, AND CAFFEINE

Recent advances in dearomatization of benzazoles, purines, and caffeine (microreview)

Microwave-Assisted Cu(I)-Catalyzed Synthesis of Unsymmetrical 1,4-Diamino-2-butynes via Cross-A3-Coupling/Decarboxylative A3-Coupling

Glyoxylic Acid: A Carboxyl Group‐Assisted Metal‐Free Decarboxylative Reaction Toward Propargylamines

Cu‐Catalyzed Selective Synthesis of Propargylamines via A3‐Coupling/Aza‐Michael Addition Sequence: Amine Loading Controls the Selectivity

Modular Synthesis of Unsymmetrical 1,4‐Diamino‐2‐butynes by Cu–Catalyzed Sequential Decarboxylative A3‐Coupling/Petasis Reaction/A3‐Coupling

Copper-catalyzed deaminative alkynylation of secondary amines with alkynes: selectivity switch in the synthesis of diverse propargylamines

CF 3 SO 3 H-enabled cascade ring-opening/dearomatization of indole derivatives to polycyclic heterocycles

铜(Ⅰ)催化丙炔酸、仲胺、醛和甲醛一锅法交叉偶联构建非对称1,4-二氨基丁炔

Ynoate-Initiated Selective C–N Esterification of Tertiary Amines under Transition-Metal and Oxidant-Free Conditions

A lysosome specific ratiometric fluorescent probe for detection of bisulfite ion based on hybrid coumarin-benzimidazolium compounds

Lewis Acid‐Free Ynoate‐Mediated Chemoselective Reduction of Carboxylic Acids to Primary Alcohols

Metal‐Free Decarboxylation of α, β‐Unsaturated Carboxylic Acids for Carbon–Carbon and Carbon–Heteroatom Coupling Reactions

DOMINO DECARBOXYLATION–CO 2 FIXATION – A ROUTE TOWARD CYCLIC CARBONATES AND OXAZOLIDINONES

Domino Decarboxylation–CO2 Fixation – a Route toward Cyclic Carbonates and Oxazolidinones (Microreview)

Synthesis of functionalized oxazolidines by multicomponent reactions of 1,2-amino alcohols (microreview)

Metal‐Free Decarboxylative A3‐Coupling/Pictet–Spengler Cascade Accessing Polycyclic Scaffolds: Propiolic Acids Exceed Alkynes

1D Fe3O4@CuSiO3 composites catalyzed decarboxylative A3-coupling for propargylamine synthesis